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8GDS image
Crystal Structure Of Rho-Associated Protein Kinase 2 (Rock2) In Complex With 4-(4-(2-(2,3-Dihydro-1H- Indol-1-Yl)-2-Oxoethyl)Phenyl)-1(2H)-Phthalazinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.71 Å Release Date: 2023-05-10
Classification: TRANSFERASE
Ligands: Z8O, SO4

7JOU image
Crystal Structure Of Rho-Associated Protein Kinase 1 (Rock1) In Complex With A Phenylpyrazole Amide Inhibitor

7JOV image
Crystal Structure Of Rho-Associated Protein Kinase 2 (Rock2) In Complex With A Phenylpyrazole Amide Inhibitor

5U6J image
Factor Viia In Complex With The Inhibitor 3-{[(2R)-17-Ethyl-4-Methyl-3,12-Dioxo-7-[(Propan-2-Yl)Sulfonyl]-13-Oxa-4,11-Diazatricyclo[14.2.2.1~6,10~]Henicosa-1(18),6(21),7,9,16,19-Hexaen-2-Yl]Amino}Benzamide

5L2Y image
Factor Viia In Complex With The Inhibitor 1-[(2R,15R)-2-[(1-Amino-4-Fluoroisoquinolin-6-Yl)Amino]-4,15,20-Trimethyl-3,12-Dioxo-13-Oxa-4,11-Diazatricyclo[14.2.2.1~6,10~]Henicosa-1(18),6,8,10(21),16,19-Hexaen-7-Yl] Cyclobutane-1-Carboxylic Acid

5L2Z image
Factor Viia In Complex With The Inhibitor 1-[(2R,15R)-2-[(1-Amino-4-Fluoroisoquinolin-6-Yl)Amino]-4,15,17-Trimethyl-3,12-Dioxo-13-Oxa-4,11-Diazatricyclo[14.2.2.1~6,10~]Henicosa-1(18),6(21),7,9,16,19-Hexaen-7-Yl]Cyclohexane-1-Carboxylic Acid

5L30 image
Factor Viia In Complex With The Inhibitor (2R,15R)-2-[(1-Aminoisoquinolin-6-Yl)Amino]-4,15,17-Trimethyl-7-[1-(1H-Tetrazol-5-Yl)Cyclopropyl]-13-Oxa-4,11-Diazatricyclo[14.2.2.1~6,10~]Henicosa-1(18),6(21),7,9,16,19-Hexaene-3,12-Dione

5I46 image
Factor Viia In Complex With The Inhibitor (2R,15R)-2-[(1-Aminoisoquinolin-6-Yl)Amino]-8-Fluoro-7-Hydroxy-4,15,17-Trimethyl-13-Oxa-4,11-Diazatricyclo[14.2.2.1~6,10~]Henicosa-1(18),6(21),7,9,16,19-Hexaene-3,12-Dione

4YT6 image
Factor Viia In Complex With The Inhibitor 4-{[(R)-[5-Ethoxy-2-Fluoro-3-(Propan-2-Yloxy)Phenyl](4-Phenyl-1H-Imidazol-2-Yl)Methyl]Amino}Benzenecarboximidamide

4YT7 image
Factor Viia In Complex With The Inhibitor 2-(2-{(R)-[(4-Carbamimidoylphenyl)Amino][5-Ethoxy-2-Fluoro-3-(Propan-2-Yloxy)Phenyl]Methyl}-1H-Imidazol-4-Yl)Benzamide

4NG9 image
Factor Viia In Complex With The Inhibitor (2R)-2-[(1-Aminoisoquinolin-6-Yl)Amino]-2-[3-Ethoxy-4-(Propan-2-Yloxy)Phenyl]-N-(3-Sulfamoylbenzyl)Ethanamide

4NGA image
Factor Viia In Complex With The Inhibitor (2R)-2-[(1-Aminoisoquinolin-6-Yl)Amino]-2-[3-Ethoxy-4-(Propan-2-Yloxy)Phenyl]-N-[2-(Propan-2-Ylsulfonyl)Benzyl]Ethanamide

4JYU image
Structure Of Factor Viia In Complex With The Inhibitor (2R)-2-[(1-Aminoisoquinolin-6-Yl)Amino]-2-[3-Ethoxy-4-(Propan-2-Yloxy)Phenyl]-N-(Phenylsulfonyl)Ethanamide

4JYV image
Structure Of Factor Viia In Complex With The Inhibitor (2R)-2-[3-Ethoxy-4-(Propan-2-Yloxy)Phenyl]-2-(Isoquinolin-6-Ylamino)-N-[(3-Sulfamoylphenyl)Sulfonyl]Ethanamide

4ISI image
Structure Of Factor Viia In Complex With The Inhibitor (6S)-N-(4-Carbamimidoylbenzyl)-1-Chloro-3-(Cyclobutylamino)-8,8-Diethyl-4-Oxo-4,6,7,8-Tetrahydropyrrolo[1,2-A]Pyrazine-6-Carboxamide

1KYJ image
Tumor Associated Mucin Motif From Cd43 Protein
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