Search Count: 16
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Cryo-Em Structure Of Human Tankyrase 2 Sam-Parp Filament Bound To Compound, Tdi-2804 (Consensus Map).
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-07-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: ZN, A1AE4 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-07-09
Ligands: ZN, A1AE4
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Cryo-Em Structure Of Human Tankyrase 2 Sam-Parp Filament Bound To Compound, Tdi-2804 (Focused Refinement Map).
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-07-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: ZN, A1AE4 |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-07-09
Ligands: ZN, A1AE4
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Cryo-Em Structure Of Human Tankyrase 2 Sam-Parp Filament Bound To Compound, Xav (Consensus Map).
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-07-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: XAV, ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-07-09
Ligands: XAV, ZN
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Cryo-Em Structure Of Human Tankyrase 2 Sam-Parp Filament Bound To Compound, Xav (Focused Refinement Map).
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-07-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: XAV, ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-07-09
Ligands: XAV, ZN
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Cryo-Em Structure Of Human Tankyrase 2 Sam-Parp Filament - Apo State (Focused Refinement Map).
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-07-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-07-09
Ligands: ZN
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Cryo-Em Structure Of Human Tankyrase 2 Sam-Parp Filament -Apo State (Consensus Map).
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2025-07-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: ZN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2025-07-09
Ligands: ZN
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Co-Crystal Structure Of Optimized Analog Tdi-13537 Provided New Insights Into The Potency Determinants Of The Sulfonamide Inhibitor Series
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2024-01-03 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: FAD, U4I, GOL |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2024-01-03
Ligands: FAD, U4I, GOL
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Cryo-Em Structure Of Mtb Lpd Bound To Inhibitor Complex With 2-((2-Cyano-N,5-Dimethyl-1H-Indole)-7-Sulfonamido)-N-(4-(Oxetan-3-Yl)-3,4-Dihydro-2H-Benzo[B] [1,4]Oxazin-7-Yl)Acetamide
Organism: Mycobacterium tuberculosis
Method: ELECTRON MICROSCOPY Release Date: 2022-05-25 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: FAD, OU6 |
Organism: Mycobacterium tuberculosis
Method: ELECTRON MICROSCOPY
Release Date: 2022-05-25
Ligands: FAD, OU6
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Macrocyclic Peptides Tdi5575 That Selectively Inhibit The Mycobacterium Tuberculosis Proteasome
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-04-28 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: U5Y, CIT, DMF |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2021-04-28
Ligands: U5Y, CIT, DMF
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Structure Of Mtb Lpd Bound To 010705
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2021-01-27 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: FAD, WPM, GOL |
Organism: Mycobacterium tuberculosis (strain atcc 25618 / h37rv)
Method: X-RAY DIFFRACTION
Release Date: 2021-01-27
Ligands: FAD, WPM, GOL
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X-Ray Co-Structure Of Rho-Associated Protein Kinase (Rock1) With A Highly Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-08-01 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: B4J, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: B4J, GOL
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X-Ray Co-Structure Of Rho-Associated Protein Kinase (Rock1) With A Highly Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-08-01 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: B4V, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: B4V, GOL
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X-Ray Co-Structure Of Rho-Associated Protein Kinase (Rock1) With A Highly Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2018-08-01 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: B4Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: B4Y
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X-Ray Co-Structure Of Rho-Associated Protein Kinase (Rock1) With A Highly Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2018-08-01 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: B5G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-01
Ligands: B5G
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X-Ray Co-Structure Of Rho-Associated Protein Kinase (Rock1) With A Potent 2H-Isoquinolin-1-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2010-12-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3NC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-08
Ligands: 3NC
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Crystal Structure Of Rho-Associated Protein Kinase (Rock1) With A Potent Isoquinolone Derivative
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2010-12-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3ND |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-08
Ligands: 3ND