Search Count: 74
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Crystal Structure Of Xiap-Bir3 With Alp2 Series Smac Mimetic Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2026-01-21 Classification: SIGNALING PROTEIN,TRANSFERASE Ligands: ZN, A1BUO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-21
Ligands: ZN, A1BUO
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Crystal Structure Of Xiap-Bir3 With Alp1 Series Smac Mimetic Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2026-01-21 Classification: SIGNALING PROTEIN Ligands: ZN, A1BVB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-21
Ligands: ZN, A1BVB
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Crystal Structure Of Ciap1-Bir3 With Xb2 Series Smac Mimetic Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-01-21 Classification: SIGNALING PROTEIN Ligands: ZN, A1BVC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-01-21
Ligands: ZN, A1BVC
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Structure Of 1 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1P
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Structure Of 5 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.00 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1R
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Structure Of 10 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:0.95 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, WYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, WYU
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Structure Of 12 In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.06 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, A1I1Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, A1I1Z
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Structure Of 18 (Bi-2493) In Complex With Gdp-Kras
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.01 Å Release Date: 2025-08-06 Classification: HYDROLASE Ligands: GDP, MG, EDO, VU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-06
Ligands: GDP, MG, EDO, VU6
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Kras G12D In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2024-10-02 Classification: ONCOPROTEIN Ligands: GCP, YLE, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GCP, YLE, MG
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Kras G12D In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2024-10-02 Classification: ONCOPROTEIN Ligands: GCP, MG, YFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GCP, MG, YFJ
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Crystal Structure Of The Brd9 Bromodomain With Bi-7189
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-06-21 Classification: GENE REGULATION Ligands: M2O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-21
Ligands: M2O
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Crystal Structure Of The Vcb Complex With Compound 1.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2023-05-31 Classification: LIGASE Ligands: WBN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-31
Ligands: WBN, CL
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Discovery Of A Kras G12V Inhibitor In Vivo Tool Compound Starting From An Hsqc-Nmr Based Fragment Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-11-09 Classification: SIGNALING PROTEIN Ligands: 2XO, GDP, MG, LX6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: 2XO, GDP, MG, LX6
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Crystal Structure Of Kras-G12C In Complex With Compound 23 (Bi-0474)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXD
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Crystal Structure Of Kras-G12C In Complex With Compound 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, MG, LXK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, MG, LXK, SO4
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Crystal Structure Of Bit-Blocked Kras-G12V-S39C In Complex With Compound 20A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-11-09 Classification: ONCOPROTEIN Ligands: GDP, 2XO, MG, LXU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: GDP, 2XO, MG, LXU
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Crystal Structure Of Compound 10 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IOD, IFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IOD, IFJ
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Crystal Structure Of Compound 6 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IFF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IFF
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Crystal Structure Of Compound 4 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2022-09-14 Classification: LIGASE Ligands: IF8, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-14
Ligands: IF8, ZN
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Crystal Structure Of Protac 5 In Complex With The Bromodomain Of Human Smarca2 And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2022-09-07 Classification: LIGASE Ligands: IEI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-09-07
Ligands: IEI
