Search Count: 14
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Egfr (T790M/V948R) In Complex With Quinazolinone Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-02-23 Classification: TRANSFERASE/Inhibitor Ligands: ANP, MG, YFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: ANP, MG, YFA
 |
Egfr Kinase (T790M/V948R) In Complex With Allosteric Inhibitor Jbj-09-063
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-09-08 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, ANP, VNS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: MG, ANP, VNS
 |
Crystal Structure Of Egfr With Mutant-Selective Dihydrodibenzodiazepinone Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-12-18 Classification: Transferase/Transferase Inhibitor Ligands: NQ1, ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: NQ1, ANP, MG
 |
Crystal Structure Of Egfr In Complex With Eai045
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-12-18 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: MG, ANP, 9LL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: MG, ANP, 9LL
 |
Egfr In Complex With A Dihydrodibenzodiazepinone Allosteric Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-12-18 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: ANP, O57, MG, AMP, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-18
Ligands: ANP, O57, MG, AMP, EDO
 |
Egfr With An Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-06-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, ANP, JBJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-05
Ligands: MG, ANP, JBJ
 |
Kras G12C In Bound To Quinazoline Based Switch Ii Pocket (Swiip) Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2017-08-23 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: GDP, MG, 91D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-23
Ligands: GDP, MG, 91D
 |
Kras G12C Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2017-08-23 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: GDP, MG, 91G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-23
Ligands: GDP, MG, 91G
 |
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, YDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, YDI
 |
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, GOL, YDK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, GOL, YDK
 |
Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2012-01-25 Classification: TRANSFERASE Ligands: YDJ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-25
Ligands: YDJ, PO4
 |
Jnk1 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-12-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, CFK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: SO4, CFK
 |
Structure-Based Design Of Protein Tyrosine Phosphatase-1B Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2005-05-04 Classification: HYDROLASE Ligands: T1D, CL, PO4, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-05-04
Ligands: T1D, CL, PO4, NA
 |
Structure-Based Design Of Protein Tyrosine Phosphatase-1B Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2005-05-04 Classification: HYDROLASE Ligands: T2D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-05-04
Ligands: T2D