Search Count: 27
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Crystal Structure Of Jak1 In Complex With Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2016-11-09 Classification: TRANSFERASE Ligands: ADP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: ADP, MG
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Crystal Structure Of Jak1 In Complex With Pf-4950736
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-11-09 Classification: transferase/transferase INHIBITOR Ligands: 6TE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 6TE
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Jak3 With Covalent Inhibitor Pf-06651600
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-11-09 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 7H4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 7H4, SO4
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Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63O |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63O
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Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63P |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63P
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Binding Site Elucidation And Structure Guided Design Of Macrocyclic Il-17A Antagonists
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-08-31 Classification: IMMUNE SYSTEM/INHIBITOR Ligands: 63Q |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: 63Q
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Covalent Inhibitor Of Lyplal1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-07-20 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 6WG, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: 6WG, NO3
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Bromo Domain Of Creb Binding Protein
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2015-10-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3OT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 3OT
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Direct Photocapture Of Bromodomains Using Tropolone Chemical Probes
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2015-10-28 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 3OT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 3OT, EDO
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Crystal Structure Of Crosslink Stabilized Long-Form Pde4B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2015-03-11 Classification: HYDROLASE Ligands: ZN, NA, MG, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: ZN, NA, MG, IOD
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Crystal Structure Of Crosslink Stabilized Long-Form Pde4B In Complex With (R)-(-)-Rolipram
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.22 Å Release Date: 2015-03-11 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, IOD, ROL, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: ZN, IOD, ROL, MG
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Structure Of Ampk In Complex With Staurosporine Inhibitor And In The Absence Of A Synthetic Activator
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.46 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor Ligands: STU, CL, SO4, AMP |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, CL, SO4, AMP
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Structure Of Ampk In Complex With Cl-A769662 Activator And Staurosporine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.34 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor/activator Ligands: STU, CL, 32J, AMP, ADP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, CL, 32J, AMP, ADP, SO4
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Structure Of Ampk In Complex With Br2-A769662Core Activator And Staurosporine Inhibitor
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.55 Å Release Date: 2014-08-06 Classification: signaling protein/inhibitor/activator Ligands: STU, 32H, CL, AMP, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-08-06
Ligands: STU, 32H, CL, AMP, SO4
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Crystal Structure Of Human Myeloperoxidase With Covalent Thioxanthine Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-03-21 Classification: OXIDOREDUCTASE Ligands: CL, 0KY, HEM, NAG, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-21
Ligands: CL, 0KY, HEM, NAG, CA
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Crystal Structure Of Apo Pbp1A From Acinetobacter Baumannii
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-12-14 Classification: Penicillin-binding protein Ligands: MES |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: MES
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Crystal Structure Of Acinetobacter Baumannii Pbp1A In Complex With Penicillin G
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-12-14 Classification: Penicillin-binding protein/ANTIBIOTIC Ligands: PNM |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: PNM
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Crystal Structure Of Acinetobacter Baumannii Pbp1A In Complex With Imipenem
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2011-12-14 Classification: PENICILLIN-BINDING PROTEIN/ANTIBIOTIC Ligands: IM2 |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: IM2
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Crystal Structure Of Acinetobacter Baumannii Pbp1A In Complex With Aztreonam
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-12-14 Classification: Penicillin-binding protein/Antibiotic Ligands: AZR |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: AZR
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Crystal Strucuture Of Acinetobacter Baumanni Pbp1A In Complex With Mc-1
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2011-12-14 Classification: Penicillin-binding protein/Antibiotic Ligands: UE1 |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: UE1
