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3QCQ image
Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-(3-Amino-1H-Indazol-6-Yl)-N4-Ethyl-2,4-Pyrimidinediamine

3QCS image
Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-[2-Amino-6-(4-Morpholinyl)-4-Pyrimidinyl]-1H-Indazol-3-Amine

3QCX image
Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 6-{2-Amino-6-[(3R)-3-Methyl-4-Morpholinyl]-4-Pyrimidinyl}-1H-Indazol-3-Amine

3QCY image
Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 4-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-N-Phenyl-2-Morpholinecarboxamide

3QD0 image
Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With (2R,5S)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-6-Methyl-N-Phenyl-3-Piperidinecarboxamide

3QD3 image
Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 1,1-Dimethylethyl {(3R,6S)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-6-Methyl-3-Piperidinyl}Carbamate

3QD4 image
Phosphoinositide-Dependent Kinase-1 (Pdk1) Kinase Domain With 1,1-Dimethylethyl{(3R,5R)-1-[2-Amino-6-(3-Amino-1H-Indazol-6-Yl)-4-Pyrimidinyl]-5-Methyl-3-Piperidinyl}Carbamate

3L54 image
Structure Of Pi3K Gamma With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2010-06-30
Classification: TRANSFERASE
Ligands: SO4, LXX

3L08 image
Structure Of Pi3K Gamma With A Potent Inhibitor: Gsk2126458
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2010-06-23
Classification: TRANSFERASE
Ligands: SO4, ZIG
Protein Functional Filters:
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