Search Count: 320
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Btk In Complex With 18A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-10-06 Classification: TRANSFERASE/INHIBITOR Ligands: 2IE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 2IE
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Btk In Complex With 25A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2021-10-06 Classification: TRANSFERASE/INHIBITOR Ligands: 2IJ, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 2IJ, DMS
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9J, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9J, DMS
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Btk1 Soaked With Compound 5, Y551 Is Sequestered
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.33 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9M
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Btk1 Soaked With Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9P, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9P, DMS
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Btk1 Soaked With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9S, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9S, DMS
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Btk1 Soaked With Compound 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: X9V, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: X9V, DMS
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Btk1 Soaked With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2021-05-19 Classification: TRANSFERASE Ligands: DMS, X9Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-19
Ligands: DMS, X9Y
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Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.13 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: QRY, CL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: QRY, CL, SO4
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Crystal Structure Of The P300 Acetyltransferase Domain With Peptide-Competitive Inhibitor 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: COA, QS4, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: COA, QS4, DMS
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Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: SO4, CL, QS1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: SO4, CL, QS1
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Crystal Structure Of The P300 Acetyltransferase Domain With Accoa Competitive Inhibitor 12
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-04-01 Classification: TRANSFERASE/INHIBITOR Ligands: QSD, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: QSD, SO4, CL
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Crystal Structure Of The P300 Acetyltransferase Domain With Allosteric Inhibitor Cpi-090 And Coa
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2019-10-23 Classification: TRANSFERASE/INHIBITOR Ligands: COA, OJ7 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: COA, OJ7
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Crystal Structure Of The P300 Acetyltransferase Domain With Allosteric Inhibitor Cpi-076 And Coa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2019-10-23 Classification: TRANSFERASE/INHIBITOR Ligands: COA, OK7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-23
Ligands: COA, OK7
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Structure Of Human Bruton'S Tyrosine Kinase In Complex With Evobrutinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2019-08-14 Classification: Transferase/Transferase Inhibitor Ligands: CL, MZJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: CL, MZJ
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Discovery Of Affinity-Based Probes For Btk Occupancy Assay
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2019-02-06 Classification: IMMUNE SYSTEM Ligands: KHD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-06
Ligands: KHD
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Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-10-17 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: GJG
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Crystal Structure Of Btk In Complex With Covalent Fragment Ligand
Organism: homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2018-10-17 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: GJD |
Organism: homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: GJD
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Crystal Structure Of Btk In Complex With Fragment Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: GJA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GJA
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Crystal Structure Of Btk In Complex With Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GJ7, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GJ7, DMS
