Search Count: 22
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Co-Crystal Structure Of Human Prmt9 In Complex With Mrk-990 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2024-12-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: A1AHM, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1AHM, UNX
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Co-Crystal Structure Of Human Carm1 In Complex With Mt556 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-01-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 44T, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-01-18
Ligands: 44T, UNX
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Co-Crystal Structure Of Human Prmt9 In Complex With Mt221 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2021-12-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EJB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-22
Ligands: EJB
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Co-Crystal Structure Of Human Prmt9 In Complex With Mt556 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-08-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 44T, EDO, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: 44T, EDO, UNX
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Co-Structure Of Btk Kinase Domain With L-005085737 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULV, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULV, 5WE
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Co-Structure Of Btk Kinase Domain With L-005191930 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULY, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULY, 5WE
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Co-Structure Of Btk Kinase Domain With L-005298385 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: UM4, EDO, BTB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: UM4, EDO, BTB
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Core Catalytic Domain Of Hiv Integrase In Complex With Virtual Screening Hit
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2020-05-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: R2D |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-05-13
Ligands: R2D
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Factor Xia In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2020-05-06 Classification: BLOOD CLOTTING Ligands: CIT, R2Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: CIT, R2Y
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Factor Xia In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2020-05-06 Classification: BLOOD CLOTTING Ligands: FLC, R3A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: FLC, R3A
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The Structure Of Dpp4 In Complex With Vildagliptin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2017-09-27 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: LF7, NAG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: LF7, NAG, NA
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The Structure Of Dpp4 In Complex With Vildagliptin Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2017-09-27 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: NAG, C8S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-27
Ligands: NAG, C8S
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Human Dpp4 In Complex With A Novel Tricyclic Hetero-Cycle Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-06-08 Classification: Hydrolase/Hydrolase Inhibitor Ligands: NAG, 6AJ, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: NAG, 6AJ, NA
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Human Dpp4 In Complex With A Novel 5,5,6-Tricyclic Pyrrolidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-05-11 Classification: Hydrolase/Hydrolase Inhibitor Ligands: NAG, NA, 6DG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-11
Ligands: NAG, NA, 6DG
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Btk-Inhibitor Co-Structure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-03-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 5WH, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-23
Ligands: 5WH, 5WE
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Btk Kinase Domain With Inhibitor 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-02-03 Classification: TRANSFERASE Ligands: 5WF, 5WE, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 5WF, 5WE, CL, EDO
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Human Dipeptidyl Peptidase Iv/Cd26 In Complex With The Long-Acting Inhibitor Omarigliptin (Mk-3102)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-04-09 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-09
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Human Dipeptidyl Peptidase Iv/Cd26 In Complex With A Novel Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-07-01 Classification: HYDROLASE Ligands: NAG, NA, 605 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-07-01
Ligands: NAG, NA, 605
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Human Dipeptidyl Peptidase 4 In Complex With A Diazepan-2-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2006-11-28 Classification: HYDROLASE Ligands: NAG, NA, 872 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
Ligands: NAG, NA, 872
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Human Dipeptidyl Peptidase 4 In Complex With A Diazepan-2-One Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2006-11-28 Classification: HYDROLASE Ligands: NAG, 565 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
Ligands: NAG, 565
