Search Count: 26
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2022-11-23 Classification: HYDROLASE Ligands: ZN, 8IY |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2022-11-02 Classification: HYDROLASE Ligands: ZN, 98O |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2022-11-02 Classification: HYDROLASE Ligands: ZN, 99I |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2022-11-02 Classification: HYDROLASE Ligands: ZN, 9DO |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-11-02 Classification: HYDROLASE Ligands: ZN, 9A1 |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2022-11-02 Classification: HYDROLASE Ligands: ZN, 9B9 |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2022-09-07 Classification: HYDROLASE Ligands: ZN, 7PX |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2022-09-07
Ligands: ZN, 7PX
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-09-07 Classification: HYDROLASE Ligands: ZN, 7PX |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-09-07 Classification: HYDROLASE Ligands: ZN, 7S6 |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2022-09-07 Classification: HYDROLASE Ligands: ZN, 7S2 |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-09-07 Classification: HYDROLASE Ligands: ZN, 7T5, EDO |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2022-09-07 Classification: HYDROLASE Ligands: ZN, 7TF |
![]() |
Lpxc Inhibitors With Fluoroproline As A Novel Zinc-Binding Group Can Serve As A Novel Class Of Antibiotic With Activity Against Multidrug-Resistant Gram-Negative Bacteria
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-09-07 Classification: HYDROLASE Ligands: ZN, 6G8 |
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2YE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2YE
![]() |
Crystal Structure Of Hpk1 In Complex With Gne1858
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F97, EDO, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: F97, EDO, MES
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2WI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2WI, SO4
![]() |
Crystal Structure Of Hpk1 In Complex With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2022-01-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 2TR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-05
Ligands: 2TR
![]() |
P110Alpha/P85Alpha With Compound 5
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-01-27 Classification: Transferase/Transferase Inhibitor Ligands: 5H2 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H2
![]() |
P110Alpha With Gdc-0326
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5, EDO
![]() |
P110Delta/P85Alpha With Gdc-0326
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.64 Å Release Date: 2016-01-27 Classification: Transferase/Inhibitor Ligands: 5H5 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: 5H5
