Search Count: 10
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Identification And Profiling Of A Selective And Brain Penetrant Radioligand For In Vivo Target Occupancy Measurement Of Casein Kinase 1 (Ck1) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2017-06-28 Classification: TRANSFERASE/INHIBITOR Ligands: 9WG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 9WG, SO4
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Crystal Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06447475)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2015-03-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MN, 3FE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: MN, 3FE
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Crystal Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06454589).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 3JA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3JA
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Structure Of Mst3 With A Pyrrolopyrimidine Inhibitor (Pf-06645342)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2015-03-18 Classification: transferase/transferase inhibitor Ligands: 3JB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3JB
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Crystal Structure Of Tyk2 In Complex With Compound 15, 6-((2,5-Dimethoxyphenyl)Thio)-3-(1-Methyl-1H-Pyrazol-4-Yl)-[1,2,4]Triazolo[4,3-B]Pyridazine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2014-09-03 Classification: TRANSFERASE Ligands: 2YK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-09-03
Ligands: 2YK
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Ck1D In Complex With 1-{4-[3-(4-Fluorophenyl)-1-Methyl-1H-Pyrazol-4-Yl]Pyridin-2-Yl}-N-Methylmethanamine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2013-09-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1QN, SO4, 1QO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 1QN, SO4, 1QO
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Ck1D In Complex With 9-[3-(4-Fluorophenyl)-1-Methyl-1H-Pyrazol-4-Yl]-2,3,4,5-Tetrahydropyrido[2,3-F][1,4]Oxazepine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2013-09-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1QM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 1QM, SO4
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Ck1D In Complex With {4-[3-(4-Fluorophenyl)-1H-Pyrazol-4-Yl]Pyridin-2-Yl}Methanol Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2013-09-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1QJ, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 1QJ, SO4, EDO
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Ck1D In Complex With (3S)-3-{4-[3-(4-Fluorophenyl)-1-Methyl-1H-Pyrazol-4-Yl]Pyridin-2-Yl}Morpholine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-09-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1QG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-18
Ligands: 1QG, SO4
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Succinic Acid Amides As P2-P3 Replacements For Inhibitors Of Interleukin-1Beta Converting Enzyme (Ice Or Caspase 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-08-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 3NS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: 3NS