Search Count: 40
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLP |
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLJ, EPE |
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Displacement Of Wdr5 From Chromatin By A Pharmacological Win Site Inhibitor With Picomolar Affinity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLS, SO4 |
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Discovery Of Potent 2-Aryl-6,7-Dihydro-5Hpyrrolo[ 1,2-A]Imidazoles As Wdr5 Win-Site Inhibitors Using Fragment-Based Methods And Structure-Based Design
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2019-03-13 Classification: gene regulation/inhibitor Ligands: HLM |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-05-31 Classification: GENE REGULATION/INHIBITOR Ligands: XKN, GOL, SO4, CL |
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Wd Repeat-Containing Protein 5 Complexed With N-[(3,5-Dimethoxyphenyl)Methyl]-4'-Fluoro-5-{[(2E)-2-Imino-3-Methyl-2,3-Dihydro-1H-Imidazol-1-Yl]Methyl}-2'-Methyl[1,1'-Biphenyl]-3-Carboxamide (Compound 13)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2020-01-01 Classification: GENE REGULATION/INHIBITOR Ligands: Q6S |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: YC4, EDO |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: Y9P, EDO |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: P2L, DMS, EDO |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: DMS, YBV, EDO |
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Crystal Structure Of The First Bromodomain Of Human Brd4 With Benzodiazepine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2021-09-01 Classification: GENE REGULATION/INHIBITOR Ligands: UDV |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2020-10-07 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, U0D |
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Crystal Structure Of Ttd-Phd Domain Of Uhrf1 In Complex With Mstella Peptide (Residues 85-119)
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2024-11-06 Classification: GENE REGULATION/INHIBITOR Ligands: ZN |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2020-01-01 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, DMS, QJ1 |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2020-01-01 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, QKD |
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Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2020-01-01 Classification: GENE REGULATION/INHIBITOR Ligands: QJA, EDO |
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Crystal Structure Of The First Bromodomain (Bd1) Of Human Brd3 Bound To Sg3-179
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2021-07-14 Classification: GENE REGULATION/INHIBITOR Ligands: 5W2, EDO, DMS |
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Crystal Structure Of The First Bromodomain (Bd1) Of Human Brd3 Bound To Erk5-In-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-07-14 Classification: GENE REGULATION/INHIBITOR Ligands: VYJ |
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Crystal Structure Of The Second Bromodomain (Bd2) Of Human Brd3 Bound To Bromosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-07-14 Classification: GENE REGULATION/INHIBITOR Ligands: BMF |
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Crystal Structure Of The First Bromodomain (Bd1) Of Human Brd2 Bound To Volasertib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2021-07-14 Classification: GENE REGULATION/INHIBITOR Ligands: IBI |