Search Count: 16
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Crystal Structure Of Human Soluble Adenylyl Cyclase (Sac) In Complex With Inhibitor Tdi-09066
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2024-01-03 Classification: SIGNALING PROTEIN Ligands: V9E, DMS, ACT, EDO, PG4, PGE, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-01-03
Ligands: V9E, DMS, ACT, EDO, PG4, PGE, CL
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Crystal Structure Of Human Soluble Adenylyl Cyclase (Sac) In Complex With Inhibitor Tdi-10512
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-04-26 Classification: SIGNALING PROTEIN Ligands: V6U, DMS, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: V6U, DMS, EDO, ACT
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Crystal Structure Of Human Soluble Adenylyl Cyclase Catalytic Domain In Complex With The Inhibitor Tdi-10228
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-04-26 Classification: SIGNALING PROTEIN Ligands: VE1, DMS, ACT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: VE1, DMS, ACT, EDO
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Complex Of Human Soluble Adenylyl Cyclase 10 Catalytic Core With Inhibitor Tdi-10962
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-04-26 Classification: SIGNALING PROTEIN Ligands: VBB, DMS, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-26
Ligands: VBB, DMS, EDO, ACT
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Crystal Structure Of Human Soluble Adenylyl Cyclase In Complex With The Inhibitor Tdi-011861
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2023-03-29 Classification: SIGNALING PROTEIN Ligands: PJU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-29
Ligands: PJU
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Human Soluble Adenylyl Cyclase In Complex With The Inhibitor Tdi10229
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2021-10-06 Classification: SIGNALING PROTEIN Ligands: 1S2, ACT, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: 1S2, ACT, DMS, EDO
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Bacterial O-Glcnacase (Oga) With Compound
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-01-13 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ACT, VUA, EDO |
Organism: Escherichia coli k-12
Method: X-RAY DIFFRACTION
Release Date: 2021-01-13
Ligands: ACT, VUA, EDO
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Halk In Complex With Compound 7 N-((1S)-1-(5-Fluoropyridin-2-Yl)Ethyl)-1-(5-Methyl-1H-Pyrazol-3-Yl)-3-(Oxetan-3-Ylsulfonyl)-1H-Pyrrolo[2,3-B]Pyridin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-05-01 Classification: PROTEIN BINDING Ligands: HKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: HKJ
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Halk In Complex With Compound 9 (6-(((1S)-1-(5-Fluoropyridin-2-Yl)Ethyl)Amino)-1-(3-Methyl-1H-Pyrazol-5-Yl)-1H-Pyrrolo[2,3-B]Pyridin-3-Yl)(Morpholin-4-Yl)Methanone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2019-05-01 Classification: TRANSFERASE/INHIBITOR Ligands: J3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: J3Y
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Halk In Complex With Compound 1 (S)-N-(1-(2,4-Difluorophenyl)Ethyl)-3-(3-Methyl-1H-Pyrazol-5-Yl)Imidazo[1,2-B]Pyridazin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-05-01 Classification: TRANSFERASE/INHIBITOR Ligands: J4M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: J4M
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Crystal Structure Of Human Monoacylglycerol Lipase In Complex With Compound 3L
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2018-10-17 Classification: HYDROLASE/INHIBITOR Ligands: 9JX, PG4, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: 9JX, PG4, EDO, CL
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Crystal Structure Of The Catalytic Domain Of Human Pde10A Complexed With N-(4-((5-Methyl-5H-Pyrrolo[3,2-D]Pyrimidin-4-Yl)Oxy)Phenyl)-1H-Benzimidazol-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2016-06-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, ZN, 6DT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: MG, ZN, 6DT
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Crystal Structure Of The Catalytic Domain Of Human Pde10A Complexed With 1-(Cyclopropylmethyl)-5-(2-(2,3-Dihydro-1H-Imidazo[1,2-A]Benzimidazol-1-Yl)Ethoxy)-3-(1-Phenyl-1H-Pyrazol-5-Yl)Pyridazin-4(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2016-06-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, ZN, 6DW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: MG, ZN, 6DW
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Crystal Structure Of The Catalytic Domain Of Pde10A Complexed With 3-(1-Phenyl-1H-Pyrazol-5-Yl)-1-(3-(Trifluoromethyl)Phenyl)Pyridazin-4(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-11-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, ZN, 3KG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: MG, ZN, 3KG
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Crystal Structure Of The Catalytic Domain Of Pde10A Complexed With 5-Methoxy-3-(1-Phenyl-1H-Pyrazol-5-Yl)-1-(3-(Trifluoromethyl)Phenyl)Pyridazin-4(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2014-11-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, 3KB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: ZN, MG, 3KB
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Crystal Structure Of The Catalytic Domain Of Pde10A Complexed With 1-(2-Fluoro-4-(1H-Pyrazol-1-Yl)Phenyl)-5-Methoxy-3-(1-Phenyl-1H-Pyrazol-5-Yl)Pyridazin-4(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-11-19 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, ZN, 3K9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: MG, ZN, 3K9