Search Count: 11
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Crystal Structure Of Cyp46A1 With [(1R,5S)-3-Oxa-8-Azabicyclo[3.2.1]Octan-8-Yl][(4R,8M)-8-(1,3-Oxazol-5-Yl)-6-(Trifluoromethyl)Imidazo[1,2-A]Pyridin-3-Yl]Methanone (Compound 3K)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2025-07-02 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BZE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-02
Ligands: HEM, A1BZE
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Crystal Structure Of Cyp46A1 With (Morpholin-4-Yl)[(4R,8M)-8-(1,3-Oxazol-5-Yl)-6-(Trifluoromethyl)Imidazo[1,2-A]Pyridin-3-Yl]Methanone (Compound 2H)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2025-07-02 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BZD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-02
Ligands: HEM, A1BZD
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Crystal Structure Of Cyp46A1 With Cyclopropyl[(4M)-4-(1,3-Oxazol-5-Yl)-6-(Trifluoromethyl)-1H-Indol-1-Yl]Methanone (Compound 2B)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2025-07-02 Classification: HYDROLASE/INHIBITOR Ligands: HEM, A1BZC, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-02
Ligands: HEM, A1BZC, EDO
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Co-Complex Cyp46A1 With 0420 (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-02-23 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: HEM, EDO, 04Y, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: HEM, EDO, 04Y, GOL
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Co-Complex Cyp46A1 With 0431 (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-02-23 Classification: HYDROLASE Ligands: HEM, 05D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-23
Ligands: HEM, 05D
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P38 In Complex With T-3220137
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-11-20 Classification: TRANSFERASE/INHIBITOR Ligands: MKP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: MKP
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[4,5-B]Pyridine-2-One Based P38 Map Kinase Inhibitors By Scaffold Hopping: Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-04-17 Classification: TRANSFERASE Ligands: J8S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: J8S
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[4,5-B]Pyridine-2-One Based P38 Map Kinase Inhibitors By Scaffold Hopping - Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-04-17 Classification: TRANSFERASE/INHIBITOR Ligands: J9G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: J9G
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Crystal Structure Of Tdr-Tdif Complex
Organism: Arabidopsis thaliana
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-08-24 Classification: SIGNALING PROTEIN Ligands: NAG |
Organism: Arabidopsis thaliana
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: NAG
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Crystal Structure Of S.A. Gyrase In Complex With Compound 7
Organism: Staphylococcus aureus, Staphylococcus aureus subsp. aureus ed98
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-06-17 Classification: Isomerase/DNA/RNA Ligands: MN, SO4, WCP |
Organism: Staphylococcus aureus, Staphylococcus aureus subsp. aureus ed98
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: MN, SO4, WCP
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Crystal Structure Of S.A. Gyrase-Am8191 Complex
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2014-06-18 Classification: ISOMERASE/ISOMERASE Inhibitor/DNA Ligands: 31N, SO4, MN |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2014-06-18
Ligands: 31N, SO4, MN