Search Count: 9
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Probing 3-Amino-2H-Azaindazoles As Allosteric Inhibitors Of The Protein Tyrosine Phosphatase Shp2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2026-06-24 Classification: PEPTIDE BINDING PROTEIN Ligands: A1JWM, ACT, EDO, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-24
Ligands: A1JWM, ACT, EDO, NA
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Il17A Homodimer Complexed To Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCE
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Il17A Complexed To Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCW, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCW, CL
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Crystal Structure Of Jak3 Complexed To N-[3-(6-Phenylamino-Pyrazin-2-Yl)-3H-Benzoimidazol-5-Yl]-Acrylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-01-14 Classification: Transferase/transferase inhibitor Ligands: 37Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-14
Ligands: 37Q
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-1,2,2-Trimethyl-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: PHU, 933 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: PHU, 933
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((S)-2-Hydroxy-1,2-Dimethyl-Propyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19Q
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((R)-2-Hydroxy-1,2-Dimethyl-Propyl
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19R
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Jak3 Kinase Domain In Complex With 2-Cyclopropyl-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid ((R)-1-Methyl-2-Oxo-2-Piperidin-1-Yl-Ethyl)-Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-01-16 Classification: Transferase/Transferase Inhibitor Ligands: 19S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-16
Ligands: 19S
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Hrxralpha & Mlxralpha With An Indole Pharmacophore, Sb786875
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2009-02-10 Classification: TRANSCRIPTION Ligands: REA, LX2 |
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2009-02-10
Ligands: REA, LX2
