Search Count: 6
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Cathepsin K Covalently Bound To A Cyano-Pyrimidine Inhibitor With Improved Selectivity Over Herg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-03-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: O47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-03-30
Ligands: O47
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Cathepsin K Covalently Bound To A 2-Cyano Pyrimidine Inhibitor With A Benzyl P3 Group.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2010-10-06 Classification: HYDROLASE Ligands: SO4, O75 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-06
Ligands: SO4, O75
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X-Ray Structure Of Cathepsin K Covalently Bound To A Triazine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: ORG, TFA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: ORG, TFA
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Cathepsin K In Complex With A Non-Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: SO4, KWZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: SO4, KWZ
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Cathepsin K In Complex With A Selective 2-Cyano-Pyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2010-03-02 Classification: HYDROLASE Ligands: KX1, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: KX1, SO4
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Cd11A (Lfa1) I-Domain Complexed With Bms-587101 Aka 5-[(5S, 9R)-9-(4-Cyanophenyl)-3-(3,5-Dichlorophenyl)-1-Methyl-2,4-Dioxo-1,3,7-Triazaspiro [4.4]Non-7-Yl]Methyl]-3-Thiophenecarboxylicacid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2006-12-19 Classification: CELL ADHESION Ligands: 2IC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-12-19
Ligands: 2IC
