Search Count: 36
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Binding Sites In The Arid1B Dna Binding Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2026-08-05 Classification: DNA BINDING PROTEIN Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: EDO
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Arid1B Arid Bound To Compound A-1 (5-(Hex-1-Yn-1-Yl)Pyridine-3-Carboxylic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.49 Å Release Date: 2026-08-05 Classification: DNA BINDING PROTEIN Ligands: A1CT6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1CT6
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Arid1B Arid Bound To Compound A-2 (5-(Hex-1-Yn-1-Yl)-3-Methylpyridin-2(1H)-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2026-08-05 Classification: DNA BINDING PROTEIN Ligands: A1CT7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1CT7
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Arid1B Arid Bound To Compound A-3 (5-(Phenylethynyl)Pyridine-3-Carboxylic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2026-08-05 Classification: DNA BINDING PROTEIN Ligands: KVD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: KVD
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Arid1B Arid Bound To Compound A-4 (N-[(5-Methylthiophen-2-Yl)Methyl]-7,8-Dihydro-5H-Pyrano[4,3-B]Pyridin-3-Amine)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2026-08-05 Classification: DNA BINDING PROTEIN Ligands: A1CT9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1CT9
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Arid1B Arid Bound To Compound B-2 ((2M)-2'-(Morpholin-4-Yl)-6-Oxo-4-(Trifluoromethyl)-1,6-Dihydro[2,3'-Bipyridine]-5-Carbonitrile)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2026-08-05 Classification: DNA BINDING PROTEIN Ligands: ZN, ACT, A1CUA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: ZN, ACT, A1CUA
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Arid1B Arid Bound To Compound C-1 (5-Fluoro-2-(1H-Pyrrolo[2,3-B]Pyridine-3-Sulfonamido)Benzoic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2026-08-05 Classification: DNA BINDING PROTEIN Ligands: A1CT8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1CT8
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Human Pi3K P85Alpha/P110Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
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P85Alpha/P110Alpha Heterodimer H1047R Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
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Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UE9
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Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UIW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UIW
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Human Pi3K P85Alpha/P110Alpha Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.53 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UIW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UIW
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Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.62 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UJC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UJC
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Human Pi3K P85Alpha/P110Alpha Bound To Rly-2608
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: XUZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: XUZ
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Cryoem Structure Of Pi3Kalpha
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-11-15 Classification: CYTOSOLIC PROTEIN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-11-15
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Tno155
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-09-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: VKS, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: VKS, PO4
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2020-09-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: VKP, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: VKP, PO4
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Idh1 R132H Mutant In Complex With Idh889
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-01-25 Classification: OXIDOREDUCTASE Ligands: FLC, 7J2, NDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: FLC, 7J2, NDP
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp836
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-07-06 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 5OA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-06
Ligands: 5OA, PO4
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Non-Receptor Protein Tyrosine Phosphatase Shp2 In Complex With Allosteric Inhibitor Shp099
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-06-29 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 5OD, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 5OD, PO4
