Search Count: 30
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Taf1-Bd2 In Complex With Cpd27 (6-(But-3-En-1-Yl)-4-(1-Methyl-6-(Morpholine-4-Carbonyl)-1H-Benzo[D]Imidazol-4-Yl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-11-14 Classification: Transcription/Inhibitor Ligands: G9V |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: G9V
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Taf1-Bd2 In Complex With Cpd8 (6-(But-3-En-1-Yl)-4-(3-(Morpholine-4-Carbonyl)Phenyl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-10-31 Classification: Transcription/Inhibitor Ligands: G9Y |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: G9Y
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Structure Of Bromodomain From Human Baz1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2017-07-12 Classification: TRANSCRIPTION Ligands: EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-07-12
Ligands: EPE
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Cecr2 In Complex With Cpd6 (6-Allyl-N,2-Dimethyl-7-Oxo-N-(1-(1-Phenylethyl)Piperidin-4-Yl)-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-06-14 Classification: Transcription/Inhibitor Ligands: SO4, 96V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-14
Ligands: SO4, 96V
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Brd9 In Complex With Cpd1 (6-Methyl-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2016-10-12 Classification: RNA BINDING PROTEIN Ligands: EDO, PEG, 67N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: EDO, PEG, 67N
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Brd9 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2016-10-12 Classification: RNA BINDING PROTEIN Ligands: 67B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 67B
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Brd9 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: 69G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 69G
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Brd4 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: 67B, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 67B, EDO, DMS
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Brd4 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: PGE, EDO, DMS, 69G, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: PGE, EDO, DMS, 69G, GOL
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Second Bromodomain Of Taf1 Bound To A Pyrrolopyridone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-06-08 Classification: PROTEIN BINDING/INHIBITOR Ligands: 67C |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 67C
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Taf1(2) Bound To A Pyrrolopyridone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.21 Å Release Date: 2016-06-08 Classification: PROTEIN BINDING/INHIBITOR Ligands: 67B, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 67B, CA
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Structure Of Histone Lysine Demethylase Kdm5A In Complex With Selective Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.14 Å Release Date: 2016-05-18 Classification: Oxidoreductase/Inhibitor Ligands: NI, ZN, 50P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: NI, ZN, 50P
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02773986
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: SCN, 68Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: SCN, 68Y
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02778174
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: EDO, SCN, 69A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: EDO, SCN, 69A
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To The Benzodiazepinone G02857790
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2016-04-20 Classification: PROTEIN BINDING/INHIBITOR Ligands: ACT, CA, 69B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ACT, CA, 69B
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Cbp In Complex With Cpd23 ((R)-6-(3-(Benzyloxy)Phenyl)-4-Methyl-1,3,4,5-Tetrahydro-2H-Benzo[B][1,4]Diazepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2016-04-20 Classification: Transcription/Protein Binding Ligands: ZN, 69F, B3P, EDO, NA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ZN, 69F, B3P, EDO, NA, PEG
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Cbp In Complex With Cpd637 ((R)-4-Methyl-6-(1-Methyl-3-(1-Methyl-1H-Pyrazol-4-Yl)-1H-Indazol-5-Yl)-1,3,4,5-Tetrahydro-2H-Benzo[B][1,4]Diazepin-2-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2016-04-20 Classification: Transcription/Protein Binding Ligands: ZN, 69E, B3P, EDO, NA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-20
Ligands: ZN, 69E, B3P, EDO, NA, PEG
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Crystal Structure Of Brd9 Bromodomain Bound To Dmso
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2015-09-16 Classification: PROTEIN BINDING Ligands: DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
Ligands: DMS
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Crystal Structure Of Brd9 Bromodomain Bound To A Butyryllysine Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2015-09-16 Classification: PROTEIN BINDING |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
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Crystal Structure Of Brd9 Bromodomain Bound To A Crotonyllysine Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2015-09-16 Classification: PROTEIN BINDING |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-16
