Search Count: 30
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Azd9291 Complex With Wild Type Egfr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-11-11 Classification: transferase/transferase inhibitor Ligands: YY3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: YY3
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1.85 Angstrom Structure Of Egfr Kinase Domain With Gefitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-11-05 Classification: transferase/transferase inhibitor Ligands: IRE, NA, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-05
Ligands: IRE, NA, MES
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1.9 Angstrom Structure Of Egfr Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-11-05 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-05
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Akr1C3 Complexed With Breakdown Product Of N-(Tert-Butyl)-2-(2-Chloro-4-(((3-Mercapto-5-Methyl-4H-1,2,4-Triazol-4-Yl)Amino)Methyl)-6-Methoxyphenoxy)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-11-05 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAP, YY2, YY1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-05
Ligands: NAP, YY2, YY1, EDO
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Akr1C2 Complex With Naproxen
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-04-02 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: NPS, NAP, EDO, TLA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: NPS, NAP, EDO, TLA, PO4
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Akr1C2 Complex With Sulindac
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2014-04-02 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: SUZ, NAP, EDO, TLA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: SUZ, NAP, EDO, TLA, PO4
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Akr1C2 Complex With Zomepirac
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2014-04-02 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: ZOM, NAP, EDO, TLA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: ZOM, NAP, EDO, TLA, PO4
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Akr1C2 Complex With Indomethacin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2014-04-02 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: IMN, NAP, TLA, EDO, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: IMN, NAP, TLA, EDO, PO4
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Akr1C2 Complex With Mefenamic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2014-04-02 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: ID8, NAP, EDO, NA, TLA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: ID8, NAP, EDO, NA, TLA, PO4
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Akr1C2 Complex With Flurbiprofen
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-04-02 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: FLP, NAP, EDO, TLA, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: FLP, NAP, EDO, TLA, PO4
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Akr1C2 Complex With Ibuprofen
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2014-04-02 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: IBP, NAP, EDO, IZP, PO4, TLA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: IBP, NAP, EDO, IZP, PO4, TLA
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With (4-(4-Chlorophenyl)Piperazin-1-Yl)(Morpholino)Methanone (24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2013-11-13 Classification: Oxidoreductase/Oxidoreductase inhibitor Ligands: NAP, 16J, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-13
Ligands: NAP, 16J, EDO
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 1-{4-[(2-Methyl-1-Piperidinyl)Sulfonyl]Phenyl}-2-Pyrrolidinone
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2013-03-20 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 10H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-20
Ligands: NAP, 10H
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W227F Active Site Mutant Of Akr1C3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-03-06 Classification: OXIDOREDUCTASE Ligands: NAP, EDO, ACT, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-03-06
Ligands: NAP, EDO, ACT, PG4
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With (R)-1-(Naphthalen-2-Ylsulfonyl)Piperidine-3-Carboxylic Acid (86)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-10-10 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: NAP, 0SL, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0SL, EDO, ACT
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 3-((3,4-Dihydroisoquinolin-2(1H)-Yl)Sulfonyl)-N-Methylbenzamide (80)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 0T0, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0T0, EDO
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Crystal Structure Of Human 17Beta-Hydroxysteroid Dehydrogenase Type 5 In Complex With 3-((3,4-Dihydroisoquinolin-2(1H)-Yl)Sulfonyl)Benzoic Acid (17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-10 Classification: oxidoreductase/oxidoreductase inhibitor Ligands: NAP, 0SZ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: NAP, 0SZ, EDO
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Akr1C3 Complex With R-Naproxen
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-08-15 Classification: OXIDOREDUCTASE Ligands: NAP, NPX, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-15
Ligands: NAP, NPX, EDO
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Akr1C3 Complex With Indomethacin At Ph 7.5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2012-08-15 Classification: OXIDOREDUCTASE Ligands: NAP, IMN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-15
Ligands: NAP, IMN, EDO
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Akr1C3 Complex With Indomethacin At Ph 6.8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2012-08-15 Classification: OXIDOREDUCTASE Ligands: NAP, IMN, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-15
Ligands: NAP, IMN, DMS, EDO