Search Count: 13
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-[6-Chloro-4-(9-Methyl-1-Oxa-4,9-Diazaspiro[5.5]Undec-4-Yl)-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl]Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2023-04-05 Classification: TRANSFERASE Ligands: XXF, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: XXF, SO4
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-{4-[(3R,5S)-3-Amino-5-Methylpiperidin-1-Yl]-6-Chloro-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3I
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With 3-{4-[(2S,5R)-5-Amino-2-Methylpiperidin-1-Yl]-6-Chloro-7H-Pyrrolo[2,3-D]Pyrimidin-5-Yl}Benzonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3O
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Pkceta Kinase Domain In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: XXF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: XXF
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Pkceta Kinase Domain In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2023-04-05 Classification: TRANSFERASE/INHIBITOR Ligands: Y3I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-04-05
Ligands: Y3I
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Crystal Structure Of Nonphosphorylated, Hpk1 Kinase Domain In Complex With Sunitinib In The Inactive State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
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Crystal Structure Of Diphosphorylated Hpk1 Kinase Domain In Complex With Sunitinib In The Active State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.97 Å Release Date: 2019-05-01 Classification: SIGNALING PROTEIN Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
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Crystal Structure Of Hpk1 Kinase Domain T165E,S171E Phosphomimetic Mutant In Complex With Sunitinib In The Inactive State.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2019-05-01 Classification: TRANSFERASE Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-01
Ligands: B49
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Wt Pcsk9-Deltac Bound To Wt Egf-A Of Ldlr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2008-11-18 Classification: HYDROLASE/RECEPTOR Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-18
Ligands: CA
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Wt Pcsk9-Deltac Bound To Egf-A H306Y Mutant Of Ldlr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-11-18 Classification: HYDROLASE/RECEPTOR Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-18
Ligands: CA
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Pcsk9-Deltac D374Y Mutant Bound To Wt Egf-A Of Ldlr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2008-11-18 Classification: HYDROLASE/RECEPTOR Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-18
Ligands: CA
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Pcsk9-Deltac D374A Mutant Bound To Wt Egf-A Of Ldlr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2008-11-18 Classification: HYDROLASE/RECEPTOR Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-18
Ligands: CA
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Pcsk9-Deltac D374H Mutant Bound To Wt Egf-A Of Ldlr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2008-11-18 Classification: HYDROLASE/RECEPTOR Ligands: CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-11-18
Ligands: CA
