Search Count: 16
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Crystal Structure Of Casein Kinase 2 (Ck2) Alpha In Complex With Bms-595
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2026-06-10 Classification: TRANSFERASE Ligands: A1DAS, MN, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: A1DAS, MN, CL
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Crystal Structure Of Kirsten Rat Sarcoma G12C Complexed With Gmppnp And Covalently Bound To An Adduct Of {(2S)-4-[7-(8-Chloronaphthalen-1-Yl)-2-{[(2S)-1-Methylpyrrolidin-2-Yl]Methoxy}-5,6,7,8-Tetrahydropyrido[3,4-D]Pyrimidin-4-Yl]-1-[(2Z)-2-Fluoro-3-(Pyridin-2-Yl)Prop-2-Enoyl]Piperazin-2-Yl}Acetonitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2025-11-05 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GNP, A1B7P, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-05
Ligands: GNP, A1B7P, MG
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Crystal Structure Of Kirsten Rat Sarcoma G12C Complexed With Gdp And Covalently Bound To An Adduct Of (2S)-1-{4-[(7P)-7-(8-Ethynyl-7-Fluoro-3-Hydroxynaphthalen-1-Yl)-8-Fluoro-2-{[(2R,4R,7As)-2-Fluorotetrahydro-1H-Pyrrolizin-7A(5H)-Yl]Methoxy}Pyrido[4,3-D]Pyrimidin-4-Yl]Piperazin-1-Yl}-2-Fluoro-3-(1,3-Thiazol-2-Yl)Propan-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-11-05 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GDP, A1B7Q, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-05
Ligands: GDP, A1B7Q, MG
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Crystal Structure Of Human Sting R232 In Complex With Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-02-09 Classification: IMMUNE SYSTEM Ligands: B7L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-09
Ligands: B7L
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7G
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7H
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7I
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-06-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-17
Ligands: Z7F
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: TKJ
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: Z7D
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Tyrosine-Protein Kinase Lck Bound To Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-10-09 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: ODJ, CXS, SO4, NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: ODJ, CXS, SO4, NI
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-{4-[3-(6-Fluoropyridin-3-Yl)-4-Oxo-4,5,6,7-Tetrahydro-1H-Pyrrolo[3,2-C]Pyridin-2-Yl]Pyridin-2-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2018-10-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2M, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: J2M, GOL
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-{4-[3-(6-Methoxypyridin-3-Yl)-1H-Pyrrolo[3,2-B]Pyridin-2-Yl]Pyridin-2-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2018-10-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: J2V
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-{4-[3-(5-Methoxypyridin-2-Yl)-1H-Pyrrolo[3,2-B] Pyridin-2-Yl]Pyridin-2-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-10-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2Y, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: J2Y, GOL
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Tgf-Beta Receptor Type 2 Kinase Domain In Complex With N- {4-[3-(6-Methoxypyridin-3-Yl)-1H-Pyrrolo[3,2-B]Pyridin-2- Yl]Pyridin-2-Yl}Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2018-10-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: J2V, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: J2V, MG, GOL
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Tgf-Beta Receptor Type 1 Kinase Domain (T204D) In Complex With N-(3-Fluoropyridin-4-Yl)-2-[6-(Trifluoromethyl)Pyridin-2-Yl]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2018-02-07 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: D0A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: D0A