Search Count: 22
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Structure Of Hdac6 Zinc-Finger Ubiquitin Binding Domain In Complex With 3-(3-(2-(Methylamino)-2-Oxoethyl)-4-Oxo-3,4-Dihydroquinazolin-2-Yl)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-05-03 Classification: HYDROLASE/INHIBITOR Ligands: ZN, ZU6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: ZN, ZU6
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Structure Of Hdac6 Zinc-Finger Ubiquitin Binding Domain In Complex With 3-(3-(2-(Benzylamino)-2-Oxoethyl)-4-Oxo-3,4-Dihydroquinazolin-2-Yl)Propanoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2023-05-03 Classification: HYDROLASE/INHIBITOR Ligands: ZN, ZU9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: ZN, ZU9
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Structure Of Hdac6 Zinc-Finger Ubiquitin Binding Domain In Complex With Sgc-Ubd253 Chemical Probe
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2023-05-03 Classification: HYDROLASE/INHIBITOR Ligands: ZN, ZUE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: ZN, ZUE
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Histone-Lysine N-Methyltransferase Nsd2-Pwwp1 With Compound Mrt10241866A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-05-05 Classification: TRANSFERASE Ligands: Y6V, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-05
Ligands: Y6V, UNX
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Histone-Lysine N-Methyltransferase Nsd2-Pwwp1 With Compound Unc6934
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: V01, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: V01, UNX
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Pwwp1 Domain Of Nsd2 In Complex With Mr837
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-11-13 Classification: TRANSFERASE Ligands: Q5D, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-13
Ligands: Q5D, UNX
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Crystal Structure Of Human Set And Mynd Domain Containing Protein 2 With Mtf9975
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-03-14 Classification: TRANSFERASE/INHIBITOR Ligands: ZN, EW4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: ZN, EW4
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Structure Of Hdac6 Zinc-Finger Ubiquitin Binding Domain Soaked With 3,3'-(Benzo[1,2-D:5,4-D']Bis(Thiazole)-2,6-Diyl)Dipropionic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: ZN, UNX, EYP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: ZN, UNX, EYP
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Crystal Structure Of Fragment 2-(Benzo[D]Thiazol-2-Yl)Acetic Acid Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: ZN, UNX, EYV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: ZN, UNX, EYV
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Crystal Structure Of Fragment 3-(Quinolin-2-Yl)Propanoic Acid Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: ZN, UNX, EYY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: ZN, UNX, EYY
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Crystal Structure Of Fragment 3-(3-Methoxy-2-Quinoxalinyl)Propanoic Acid Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: ZN, UNX, EY7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: ZN, UNX, EY7
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Crystal Structure Of Fragment 3-(3-Methyl-4-Oxo-3,4-Dihydroquinazolin-2-Yl)Propanoic Acid Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: ZN, EYA, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: ZN, EYA, UNX
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Crystal Structure Of Fragment 3-(1-Methyl-2-Oxo-1,2-Dihydroquinoxalin-3-Yl)Propionic Acid Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: ZN, EYM, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: ZN, EYM, UNX
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Crystal Structure Of Fragment 3-(1,3-Benzothiazol-2-Yl)Propanoic Acid Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: ZN, UNX, EYJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: ZN, UNX, EYJ
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Crystal Structure Of Fragment 3-(3-(Pyridin-2-Ylmethoxy)Quinoxalin-2-Yl)Propanoic Acid Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2017-08-23 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, B8P, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-23
Ligands: ZN, B8P, UNX
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Crystal Structure Of Fragment 3-(3-Benzyl-2-Oxo-2H-[1,2,4]Triazino[2,3-C]Quinazolin-6-Yl)Propanoic Acid Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2017-08-02 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 9ZV, UNX, FMT, CL, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-02
Ligands: ZN, 9ZV, UNX, FMT, CL, ACT
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Crystal Structure Of Setdb1 Tudor Domain In Complex With Fragment Mrt0181A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-08-03 Classification: Transcription/Transcription Inhibitor Ligands: 6S5, BME, SO4, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-03
Ligands: 6S5, BME, SO4, UNX
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Crystal Structure Of A Low Occupancy Fragment Candidate (N-(4-Methyl-1,3-Thiazol-2-Yl)Propanamide) Bound Adjacent To The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2016-07-27 Classification: HYDROLASE Ligands: ZN, FMT, 6T4, UNX, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-27
Ligands: ZN, FMT, 6T4, UNX, NA
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Crystal Structure Of Fragment (3-(5-Chloro-1,3-Benzothiazol-2-Yl)Propanoic Acid) Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-07-27 Classification: HYDROLASE Ligands: ZN, UNX, 6U6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-27
Ligands: ZN, UNX, 6U6
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Crystal Structure Of Fragment (3-[6-Oxo-3-(3-Pyridinyl)-1(6H)-Pyridazinyl]Propanoic Acid) Bound In The Ubiquitin Binding Pocket Of The Hdac6 Zinc-Finger Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-07-27 Classification: HYDROLASE Ligands: ZN, 6T7, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-27
Ligands: ZN, 6T7, UNX
