Search Count: 15
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Discovery Of Imidazoquinolines As A Novel Class Of Potent, Selective And In Vivo Efficacious Cot Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-08-24 Classification: TRANSFERASE Ligands: 6DA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-24
Ligands: 6DA
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Crystal Structure Of Cot Kinase Domain In Complex With 5-(2-Amino-5-(Quinolin-3-Yl)Pyridin-3-Yl)-1,3,4-Oxadiazole-2(3H)-Thione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2015-05-06 Classification: TRANSFERASE Ligands: 49B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 49B
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Crystal Structure Of Cot Kinase Domain In Complex With 5-(5-(1H-Indol-3-Yl)-1H-Pyrrolo[2,3-B]Pyridin-3-Yl)-1,3,4-Oxadiazol-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2015-05-06 Classification: TRANSFERASE Ligands: 499 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-05-06
Ligands: 499
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Abl Kinase In Complex With Imatinib And A Fragment (Frag1) In The Myristate Pocket
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-05-26 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: STI, MS9, CL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-05-26
Ligands: STI, MS9, CL
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Abl Kinase In Complex With Imatinib And Fragment (Frag2) In The Myristate Site
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: STI, MS7 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-05-26
Ligands: STI, MS7
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Structure Of Abl Kinase In Complex With Imatinib And Gnf-2
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2010-01-19 Classification: TRANSFERASE Ligands: STJ, STI, CL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-01-19
Ligands: STJ, STI, CL
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Human Abl Kinase In Complex With Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2008-04-22 Classification: TRANSFERASE Ligands: NIL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-22
Ligands: NIL
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The Crystal Structure Of The Kinase Domain Of The Protein Kinase C Theta In Complex With Nvp-Xaa228 At 2.32A Resolution.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2008-02-05 Classification: TRANSFERASE Ligands: LG8, MPD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-05
Ligands: LG8, MPD
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Human Abl Kinase Domain In Complex With Imatinib (Sti571, Glivec)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: STI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: STI
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Abl Kinase Domain In Complex With Nvp-Aeg082
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: GIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: GIN
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Abl Kinase Domain Unligated And In Complex With Tetrahydrostaurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: 4ST |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: 4ST
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Abl Kinase Domain In Complex With Pd180970
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: JIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: JIN
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Abl Kinase Domain In Complex With Nvp-Afg210
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2007-01-16 Classification: TRANSFERASE Ligands: KIN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2007-01-16
Ligands: KIN
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Structure Of Unphosphorylated C-Src In Complex With An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2005-06-21 Classification: TRANSFERASE Ligands: SO4, MPZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-06-21
Ligands: SO4, MPZ
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Kallikrein Complexed With Hirustasin
Organism: Sus scrofa, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 1997-12-24 Classification: COMPLEX (PROTEASE/INHIBITOR) |
Organism: Sus scrofa, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 1997-12-24