Search Count: 25
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Crystal Structure Of Cdk2 Bound By Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1INI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1INI
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Crystal Structure Of Cdk2-Cyclin E1 Bound By Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1IOI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1IOI
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Crystal Structure Of Cdk2-Cyclin E1 Bound By Compound 11 (Azd8421)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-09-10 Classification: TRANSFERASE Ligands: A1IOP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1IOP
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITC
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITA
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Crystal Structure Of Hpk1 T165E/S171E In Complex With Pyrazine Carboxamide Inhibitor Az3246 (Compound 24)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2025-02-19 Classification: TRANSFERASE Ligands: A1ITB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1ITB, EDO
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
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Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNE
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNH
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Oestrogen Receptor Ligand Binding Domain In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNK
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Human Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2020-04-29 Classification: TRANSFERASE Ligands: LKT, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: LKT, EDO
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Human Jak1 Kinase Domain In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-04-29 Classification: TRANSFERASE Ligands: LKQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: LKQ
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Crystal Structure Of The A2A-Star2-Bril562 In Complex With Azd4635 At 2.0A Resolution
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-06-26 Classification: MEMBRANE PROTEIN |
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
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Induced Myeloid Leukemia Cell Differentiation Protein Fabcomplex In Complex With Azd5991
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-12-26 Classification: APOPTOSIS Ligands: E4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4W
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Mcl1 In Complex With An Indole Acid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-12-26 Classification: IMMUNE SYSTEM Ligands: E4Q, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4Q, EDO
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Mcl1 In Complex With Indole Acid Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-12-26 Classification: IMMUNE SYSTEM Ligands: E4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-12-26
Ligands: E4K
