Search Count: 24
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Smarca2 In Complex With A Pyridine-2-One-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2025-04-09 Classification: DNA BINDING PROTEIN Ligands: ADP, A1AHQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-09
Ligands: ADP, A1AHQ
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Crystal Structure Of Setd2 Bound To An Indole-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2022-08-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAM, KS6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: ZN, SAM, KS6
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Crystal Structure Of Setd2 Bound To An Indole-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-08-31 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SAM, KRF, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: ZN, SAM, KRF, EDO
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Crystal Structure Of Setd2 Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-09-22 Classification: TRANSFERASE Ligands: ZN, SAM, YJ1, BME |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: ZN, SAM, YJ1, BME
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Crystal Structure Of Setd2 Bound To Compound 35
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-09-22 Classification: TRANSFERASE Ligands: ZN, SAM, YHY, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: ZN, SAM, YHY, EDO, DMS
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Crystal Structure Of Setd2 Bound To Compound 57
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2021-09-22 Classification: TRANSFERASE Ligands: ZN, SAM, YHV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-22
Ligands: ZN, SAM, YHV, EDO
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X-Ray Structure Of Mmp-13 In Complex With 4-(1,2,3-Thiadiazol-4-Yl)Pyridine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-08-04 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, 9DY, FMT, PGE, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-04
Ligands: ZN, CA, 9DY, FMT, PGE, PG4
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Il36R Extracellular Domain In Complex With Bi655130 Fab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2020-04-22 Classification: CYTOKINE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-22
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X-Ray Structure Of Nuclear Receptor Ror-Gammat Ligand Binding Domain + Src2 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2017-06-07 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
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X-Ray Co-Structure Of Nuclear Receptor Ror-Gammat Ligand Binding Domain With An Inverse Agonist And Src2 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2017-06-07 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
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X-Ray Co-Structure Of Nuclear Receptor Ror-Gammat Ligand Binding Domain With An Inverse Agonist And Src2 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2017-06-07 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
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X-Ray Co-Structure Of Nuclear Receptor Ror-Gammat Ligand Binding Domain With An Agonist And Src2 Peptide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.34 Å Release Date: 2017-06-07 Classification: TRANSCRIPTION |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
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Crystal Structure Of Human Growth Differentiation Factor 11 (Gdf-11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2016-03-09 Classification: HORMONE Ligands: PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-03-09
Ligands: PG4
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X-Ray Co-Structure Of Mmp-13 With Ethyl 5-Carbamoyl-1H-Indole-2-Carboxylate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-06-17 Classification: Hydrolase/Hydrolase inhibitor Ligands: 4UM, ZN, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: 4UM, ZN, CA
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X-Ray Co-Structure Of Mmp-13 With Ethyl 5-(1-Methyl-1H-Imidazol-5-Yl)-1H-Indole-2-Carboxylate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-06-17 Classification: Hydrolase/Hydrolase inhibitor Ligands: ZN, CA, 4UE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: ZN, CA, 4UE
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X-Ray Co-Structure Of Mmp-13 With 4-[({5-[2-(Ethoxycarbonyl)-1H-Indol-5-Yl]-1-Methyl-1H-Pyrazol-3-Yl}Formamido)Methyl]Benzoate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2015-06-17 Classification: Hydrolase/Hydrolase inhibitor Ligands: ZN, CA, 4UF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: ZN, CA, 4UF
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Crystal Structure Of Human Chymase With Benzimidazolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2011-07-20 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, ZN, 0BB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-07-20
Ligands: NAG, ZN, 0BB
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Soluble Epoxide Hydrolase In Complex With Pyrazole Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2010-10-27 Classification: HYDROLASE Ligands: MZL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-10-27
Ligands: MZL
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Crystal Structure Of Soluble Epoxide Hydrolase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.79 Å Release Date: 2010-04-28 Classification: HYDROLASE Ligands: 24D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-28
Ligands: 24D
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Crystal Structure Of Soluble Epoxide Hydrolase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2009-10-13 Classification: HYDROLASE Ligands: 33N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-13
Ligands: 33N
