Search Count: 17
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Crystal Structure Of Sars-Cov-2 Mpro With Ab-343.
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2024-12-04 Classification: VIRAL PROTEIN Ligands: A1IMY, CL, PEG, EDO |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1IMY, CL, PEG, EDO
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Crystal Structure Of Sars-Cov-2 Mpro With Compound 5
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1IL0 |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1IL0
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Crystal Structure Of Sars-Cov-2 Mpro With Compound 12
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-11-06 Classification: HYDROLASE Ligands: A1IL7, SO4, GOL, EDO |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-11-06
Ligands: A1IL7, SO4, GOL, EDO
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Hbv Capsid With Compound 3I
Organism: Hepatitis b virus
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2024-09-25 Classification: VIRAL PROTEIN Ligands: A1AVK |
Organism: Hepatitis b virus
Method: X-RAY DIFFRACTION
Release Date: 2024-09-25
Ligands: A1AVK
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Hbv Capsid Y132A With Compound 10B At 2.5A Resolution
Organism: Hepatitis b virus genotype a
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2022-05-04 Classification: VIRAL PROTEIN/INHIBITOR Ligands: 8EI |
Organism: Hepatitis b virus genotype a
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: 8EI
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Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y4
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Brain Penetrant Liver X Receptor (Lxr) Modulators Based On A 2,4,5,6-Tetrahydropyrrolo[3,4-C]Pyrazole Core
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-09-21 Classification: DNA BINDING PROTEIN Ligands: 6Y8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-21
Ligands: 6Y8
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Discovery Of Novel, Orally Efficacious Liver X Receptor (Lxr) Beta Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2016-06-29 Classification: DNA BINDING PROTEIN Ligands: 67S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-29
Ligands: 67S
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Potent And Selective Phosphodiesterase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2012-09-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: ZN, MG, 0T7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-05
Ligands: ZN, MG, 0T7
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Potent And Selective Phosphodiesterase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2012-09-05 Classification: Hydrolase/Hydrolase inhibitor Ligands: ZN, MG, 0T6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-05
Ligands: ZN, MG, 0T6
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Highly Potent, Selective, And Orally Active Phosphodiestarase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CL, 540, ZN, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: CL, 540, ZN, MG
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Highly Potent, Selective, And Orally Active Phosphodiestarase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, CL, 546 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: ZN, MG, CL, 546
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Highly Potent, Selective, And Orally Active Phosphodiestarase 10A Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2011-10-26 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, MG, 548 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: ZN, MG, 548
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Pyrazolyl And Thienyl Aminohydantoins As Potent Bace1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 591 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: 591
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Pyrazolyl And Thienyl Aminohydantoins As Potent Bace1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2011-08-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 532 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-31
Ligands: 532
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X-Ray Structure Of Bace-1 In Complex With Compound 3.B.10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-12-09 Classification: HYDROLASE Ligands: 310 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-09
Ligands: 310
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X-Ray Structure Of Bace-1 In Complex With Compound 6G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-12-09 Classification: HYDROLASE Ligands: 411 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-09
Ligands: 411
