Search Count: 32
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Pqr530 [(S)-4-(Difluoromethyl)-5-(4-(3-Methylmorpholino)-6-Morpholino-1,3,5-Triazin-2-Yl)Pyridin-2-Amine] Bound To The Pi3Ka Catalytic Subunit P110Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2019-06-26 Classification: TRANSFERASE Ligands: M1J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: M1J
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Waap In Complex With Acyl Carrier Protein
Organism: Pseudomonas aeruginosa, Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-04-03 Classification: HYDROLASE Ligands: G9S |
Organism: Pseudomonas aeruginosa, Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2019-04-03
Ligands: G9S
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Abl1 In Complex With Compound 7 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: GOL, CL, FYW, STI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: GOL, CL, FYW, STI
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Abl1 In Complex With Compound6 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-09-12 Classification: TRANSFERASE Ligands: CL, FYH, STI |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2018-09-12
Ligands: CL, FYH, STI
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Pqr309 - A Potent, Brain-Penetrant, Orally Bioavailable, Pan-Class I Pi3K/Mtor Inhibitor As Clinical Candidate In Oncology
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-09-06 Classification: TRANSFERASE Ligands: A3W, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-06
Ligands: A3W, SO4
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Tubulin Mtd265-R1 Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-03-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GOL, UGI, GDP, MES, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-03-22
Ligands: GTP, MG, CA, GOL, UGI, GDP, MES, ACP
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Structure Of Phosphoinositide 3-Kinase Gamma (Pi3K) Bound To The Potent Inhibitor Pikin2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2017-03-15 Classification: TRANSFERASE Ligands: 6K7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 6K7, SO4
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Structure Of Phosphoinositide 3-Kinase Gamma (Pi3K) Bound To The Potent Inhibitor Pikin3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-03-15 Classification: TRANSFERASE Ligands: 6K5, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-15
Ligands: 6K5, SO4
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Tubulin-Bkm120 Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2017-02-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GOL, GDP, MES, SD5, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: GTP, MG, CA, GOL, GDP, MES, SD5, ACP
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Tubulin-Mtd147 Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-02-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GOL, FB7, GDP, MES, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: GTP, MG, CA, GOL, FB7, GDP, MES, ACP
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Tubulin-Mtd265 Complex
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2017-02-22 Classification: CELL CYCLE Ligands: GTP, MG, CA, GOL, 918, GDP, MES, ACP |
Organism: Rattus norvegicus, Gallus gallus, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-02-22
Ligands: GTP, MG, CA, GOL, 918, GDP, MES, ACP
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Serine/Threonine-Protein Kinase Pak1 Complexed With A Dibenzodiazepine: Identification Of An Allosteric Site On Pak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-05 Classification: Transferase/transferase inhibitor Ligands: 4PV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4PV, GOL
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Pak1 In Complex With 2-Chloro-5-Ethyl-8-Fluoro-11-(4-Methylpiperazin-1-Yl)-Dibenzodiazepine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OQ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OQ, MG
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Pak1 In Complex With (S)-N-(Tert-Butyl)-3-((2-Chloro-5-Ethyl-8-Fluoro-Dibenzodiazepin-11-Yl)Amino)Pyrrolidine-1-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-06-24 Classification: TRANSFERASE Ligands: 4OR, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
Ligands: 4OR, MG
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Co-Crystal Structures Of The Lipid Kinase Pi3K Alpha With Pan And Isoform Selective Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SCN, 1LT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: SCN, 1LT
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Crystal Structure Of Pi3K Gamma With 5-(2,4-Dimorpholinopyrimidin-6-Yl)-4-(Trifluoromethyl)Pyridin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2012-01-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SD5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-04
Ligands: SD5
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Abl Kinase In Complex With Imatinib And A Fragment (Frag1) In The Myristate Pocket
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2010-05-26 Classification: TRANSFERASE/TRANSFERASE REGULATOR Ligands: STI, MS9, CL |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-05-26
Ligands: STI, MS9, CL
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Abl Kinase In Complex With Imatinib And Fragment (Frag2) In The Myristate Site
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2010-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: STI, MS7 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-05-26
Ligands: STI, MS7
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Crystal Structure Of The Human Clk3 In Complex With Dki
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2009-10-20 Classification: TRANSFERASE Ligands: DKI, SO4, DMS, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-20
Ligands: DKI, SO4, DMS, EDO, CL
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Crystal Structure Of The Human Clk3 In Complex With V25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2009-10-20 Classification: TRANSFERASE Ligands: V25, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-20
Ligands: V25, SO4, CL