Search Count: 28
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Crystal Structure Of Cbl-B Tkb Bound To Compound 26
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2024-07-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, A1AEG, GOL, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, A1AEG, GOL, PEG
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Crystal Structure Of Cbl-B Tkb Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2024-07-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, CA, A1AD4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, CA, A1AD4
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Crystal Structure Of Braf Kinase Domain Bound To Gdc0879
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2022-10-26 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 29L, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-26
Ligands: 29L, CL
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Crystal Structure Of Apo Egfr Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2022-10-26 Classification: TRANSFERASE Ligands: MES, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-26
Ligands: MES, SO4
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Structure Of Ciap With Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-11-18 Classification: LIGASE Ligands: ZN, TKY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: ZN, TKY
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Ternary Complex Structure - Btk Ciap Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2020-11-18 Classification: LIGASE/TRANSFERASE Ligands: TL7, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: TL7, ZN
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Ternary Complex Structure - Btk Ciap Compound 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.80 Å Release Date: 2020-11-18 Classification: LIGASE/TRANSFERASE Ligands: TKY, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-18
Ligands: TKY, ZN
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Human Immunoproteasome 20S Particle In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2019-09-11 Classification: HYDROLASE Ligands: SCN, NA, HUJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-11
Ligands: SCN, NA, HUJ
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P110Delta/P85Alpha With Taselisib (Gdc-0032)
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2017-01-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 799 |
Organism: Homo sapiens, Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 799
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Imidazobenzoxepin Compound 3
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: SO4, 76Z |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, 76Z
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Benzoxepin Compound 2
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: 774, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 774, SO4
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Crystal Structure Of Murine Nf-Kappab Inducing Kinase (Nik) Bound To Aryl Pyrrole Fragment 17
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2017-01-11 Classification: TRANSFERASE Ligands: SO4, 76Y |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: SO4, 76Y
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Crystal Structure Of Tubulin-Stathmin-Ttl-Compound 11 Complex
Organism: Rattus norvegicus, Gallus gallus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-12-28 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: GTP, MG, CA, GDP, 6YK, ADP |
Organism: Rattus norvegicus, Gallus gallus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: GTP, MG, CA, GDP, 6YK, ADP
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Jak2 Kinase (Jh1 Domain) Mutant P1057A In Complex With Tg101209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2016-11-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, ZN, 1M3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: CL, ZN, 1M3
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Discovery Of Cytotoxic Dolastatin 10 Analogs With N-Terminal Modifications
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:3.11 Å Release Date: 2015-03-25 Classification: STRUCTURAL PROTEIN/INHIBITOR Ligands: GTP, MG, GDP, LOC, 3WD |
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GTP, MG, GDP, LOC, 3WD
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Discovery Of Cytotoxic Dolastatin 10 Analogs With N-Terminal Modifications
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2015-03-25 Classification: Structural Protein/Inhibitor Ligands: GTP, MG, GDP, LOC, 3WZ |
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GTP, MG, GDP, LOC, 3WZ
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Discovery Of Cytotoxic Dolastatin 10 Analogs With N-Terminal Modifications
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:3.19 Å Release Date: 2015-03-25 Classification: Structural Protein/Inhibitor Ligands: GTP, MG, GDP, LOC, 3WV |
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GTP, MG, GDP, LOC, 3WV
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Discovery Of Cytotoxic Dolastatin 10 Analogs With N-Terminal Modifications
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2015-03-25 Classification: Structural Protein/Inhibitor Ligands: GTP, MG, GDP, LOC, 3WY |
Organism: Rattus norvegicus, Ovis aries
Method: X-RAY DIFFRACTION
Release Date: 2015-03-25
Ligands: GTP, MG, GDP, LOC, 3WY
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Crystal Structure Of Rorc In Complex With A Phenyl Sulfonamide Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-01-14 Classification: TRANSCRIPTION Ligands: 3SN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-14
Ligands: 3SN
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Crystal Structure Of Rorc In Complex With A Benzyl Sulfonamide Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2015-01-14 Classification: TRANSCRIPTION Ligands: 3SX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-14
Ligands: 3SX, SO4
