Search Count: 47
![]() |
Crystal Structure Of Compound 3-Mediated Ternary Complex Of Kras G12V C118S Gdp With Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2025-11-12 Classification: ONCOPROTEIN Ligands: A1JH1, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1JH1, GDP, MG
![]() |
Crystal Structure Of Acbi4-Mediated Ternary Complex Of Kras G12D C118S Gdp With Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2025-11-12 Classification: ONCOPROTEIN Ligands: A1JHI, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1JHI, GDP, MG
![]() |
Crystal Structure Of Compound 1-Mediated Ternary Complex Of Kras G12R Gcp With Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2025-11-12 Classification: ONCOPROTEIN Ligands: GOL, X53, GCP, MG, FLC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: GOL, X53, GCP, MG, FLC
![]() |
Crystal Structure Of Compound 3-Mediated Ternary Complex Of Kras G12R Gcp With Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2025-11-12 Classification: ONCOPROTEIN Ligands: FLC, A1JH1, GCP, MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: FLC, A1JH1, GCP, MG, GOL
![]() |
Crystal Structure Of Acbi4-Mediated Ternary Complex Of Kras G12R Gcp With Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2025-11-12 Classification: ONCOPROTEIN Ligands: SO4, A1JHI, GCP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: SO4, A1JHI, GCP, MG
![]() |
Kras G12D In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.16 Å Release Date: 2024-10-02 Classification: ONCOPROTEIN Ligands: GCP, YLE, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GCP, YLE, MG
![]() |
Kras G12D In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.31 Å Release Date: 2024-10-02 Classification: ONCOPROTEIN Ligands: GCP, MG, YFJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GCP, MG, YFJ
![]() |
Protac-Mediated Complex Of Kras With Vhl/Elongin-B/Elongin-C/Cullin-2/Rbx1
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.50 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: ZN, GDP, WYL |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-12-06
Ligands: ZN, GDP, WYL
![]() |
Kras-G12C In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2023-12-06 Classification: TRANSFERASE Ligands: GDP, MG, WYU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: GDP, MG, WYU
![]() |
Crystal Structure Of Ligand Acbi3 In Complex With Kras G12D C118S Gdp And Pvhl:Elonginc:Elonginb Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2023-12-06 Classification: GENE REGULATION Ligands: PO4, WYL, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: PO4, WYL, GDP, MG
![]() |
Crystal Structure Of Compound 3 In Complex With Kras G12V C118S Gdp And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2023-12-06 Classification: ONCOPROTEIN Ligands: GDP, X4R, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: GDP, X4R, MG
![]() |
Crystal Structure Of Compound 4 In Complex With Kras G12V C118S Gdp And Pvhl:Elonginc:Elonginb
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2023-12-06 Classification: ONCOPROTEIN Ligands: X53, GDP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: X53, GDP, MG
![]() |
Her2 In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2022-07-27 Classification: TRANSFERASE Ligands: 70I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-27
Ligands: 70I
![]() |
Crystal Structure Of Sos1 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-03-24 Classification: PROTEIN BINDING Ligands: S2Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: S2Q
![]() |
Crystal Structure Of Sos1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2021-03-24 Classification: PROTEIN BINDING Ligands: IMD, S2Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: IMD, S2Z
![]() |
Crystal Structure Of Sos1 In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2021-03-24 Classification: PROTEIN BINDING Ligands: IMD, S3Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: IMD, S3Q
![]() |
Crystal Structure Of Sos1 In Complex With Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-03-24 Classification: PROTEIN BINDING Ligands: IMD, S3T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: IMD, S3T
![]() |
Crystal Structure Of Sos1 In Complex With Compound 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-03-24 Classification: PROTEIN BINDING Ligands: IMD, S3Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: IMD, S3Z
![]() |
Crystal Structure Of Sos1 In Complex With Compound 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2021-03-24 Classification: PROTEIN BINDING Ligands: IMD, S2W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: IMD, S2W
![]() |
Sos1 In Complex With Inhibitor Bi-3406
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2020-08-26 Classification: ONCOPROTEIN Ligands: IMD, EDO, L7H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: IMD, EDO, L7H
