Search Count: 5
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Egfr Kinase Domain In Complex With Mutant Selective Allosteric Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2016-06-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, ANP, 57N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: MG, ANP, 57N
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Crystal Structure Of Egfr 696-1022 L858R In Complex With Fiin-3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2014-11-12 Classification: TRANSFERASE Ligands: FI3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-12
Ligands: FI3
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Crystal Structure Of Fgf Receptor (Fgfr) 4 Kinase Domain In Complex With Fiin-2, An Irreversible Tyrosine Kinase Inhibitor Capable Of Overcoming Fgfr Kinase Gate-Keeper Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-10-29 Classification: Transferase/transferase inhibitor Ligands: 37O, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-29
Ligands: 37O, SO4
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Crystal Structure Of Fgf Receptor (Fgfr) 4 Kinase Harboring The V550L Gate-Keeper Mutation In Complex With Fiin-3, An Irreversible Tyrosine Kinase Inhibitor Capable Of Overcoming Fgfr Kinase Gate-Keeper Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2014-10-29 Classification: Transferase/transferase inhibitor Ligands: FI3, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-29
Ligands: FI3, SO4
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Crystal Structure Of Egfr 696-1022 T790M Mutant Covalently Binding To Wz4002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-01-12 Classification: TRANSFERASE Ligands: 0UN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: 0UN
