Search Count: 5
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Discovery Of Novel, Dual Mechanism Erk Inhibitors By Affinity Selection Screening Of An Inactive Kinase State
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2014-11-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3G7, SO4 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2014-11-12
Ligands: 3G7, SO4
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P38Alpha Bound To Novel Dgf-Out Compound Pf-00215955
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2009-11-17 Classification: TRANSFERASE Ligands: JZJ, I46 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-17
Ligands: JZJ, I46
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P38Alpha Bound To Novel Dfg-Out Compound Pf-00416121
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: F4C, I46 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: F4C, I46
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Kit Kinase Domain In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: B49 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: B49
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Kit Kinase Domain Mutant D816H In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-02-24 Classification: TRANSFERASE Ligands: B49, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-02-24
Ligands: B49, SO4
