Search Count: 16
![]() |
Crystal Structure Of Khk-C And Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2023-12-06 Classification: SUGAR BINDING PROTEIN Ligands: WNH, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: WNH, SO4, GOL
![]() |
Crystal Structure Of Khk-C And Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2023-12-06 Classification: SUGAR BINDING PROTEIN Ligands: WRE, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-06
Ligands: WRE, SO4, GOL
![]() |
The Co-Crystal Structure Of Low Molecular Weight Protein Tyrosine Phosphatase (Lmw-Ptp) With A Small Molecule Inhibitor Spaa-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-10-19 Classification: HYDROLASE Ligands: OIF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-19
Ligands: OIF
![]() |
Crystal Structure Of Aicarft Bound To An Antifolate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2018-01-10 Classification: TRANSFERASE, HYDROLASE Ligands: 8UM, AMZ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-10
Ligands: 8UM, AMZ, MG
![]() |
Crystal Structure Of Aicarft Bound To An Antifolate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2018-01-10 Classification: TRANSFERASE, HYDROLASE Ligands: AMZ, MG, 8US |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-10
Ligands: AMZ, MG, 8US
![]() |
Bace Crystal Structure With Hydroxy Pyrrolidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2017-11-15 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: DJS, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: DJS, GOL
![]() |
Bace Crystal Structure With Hydroxy Pyrrolidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2017-11-15 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: DJV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: DJV, GOL
![]() |
Bace Crystal Structure With Hydroxy Morpholine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2017-11-15 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: DK7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: DK7, GOL
![]() |
Bace Crystal Structure With Hydroxy Pyrrolidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2017-11-15 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: DKJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: DKJ, GOL
![]() |
Crystal Structure Of Insulin Degrading Enzyme Complexed With Inhibitor Tert-Butyl [(2S)-2-(2,5-Difluorophenyl)-3-(Quinolin-3-Yl)Propyl]Carbamate
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2015-06-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2PJ, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: 2PJ, ZN
![]() |
Crystal Structure Of Insulin Degrading Enzyme Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2015-06-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2QW, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: 2QW, ZN
![]() |
Crystal Structure Of Insulin Degrading Enzyme Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-06-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: 2Q6, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: 2Q6, ZN
![]() |
Crystal Structure Of Insulin Degrading Enzyme Complexed With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2015-06-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 2QX, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: 2QX, ZN
![]() |
Crystal Structure Of Human Adamts-4 In Complex With Inhibitor (Compound 1, 2-(4-Chlorophenoxy)-N-{[(4R)-4-Methyl-2,5-Dioxoimidazolidin-4-Yl]Methyl} Acetamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.24 Å Release Date: 2014-12-10 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, 3PQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: ZN, CA, 3PQ
![]() |
Crystal Structure Of Human Adamts-4 In Complex With Inhibitor 5-Chloro-N-{[(4R)-2,5-Dioxo-4-(1,3-Thiazol-2-Yl)Imidazolidin-4-Yl]Methyl}-1-Benzofuran-2-Carboxamide (Compound 10)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2014-12-10 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, EDO, 3PU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: ZN, CA, EDO, 3PU
![]() |
Crystal Structure Of Human Adamts-4 In Complex With Inhibitor 5-Chloro-N-{[(4S)-4-(1-Methyl-1H-Imidazol-2-Yl)-2,5-Dioxoimidazolidin-4-Yl]Methyl}-1-Benzofuran-2-Carboxamide (Compound 11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2014-12-10 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, CA, EDO, 3PW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-10
Ligands: ZN, CA, EDO, 3PW
