Structural Entry Filters:

Search Count: 18

Download
9O63 image
Crystal Structure Of Plk4 And Rp1664 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.26 Å Release Date: 2025-05-28
Classification: TRANSFERASE
Ligands: SO4, A1CAD

7TAB image
G-925 Bound To The Smarca4 (Brg1) Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.16 Å Release Date: 2022-08-17
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: GGU

7TD9 image
G-059 Bound To The Smarca4 (Brg1) Bromodomain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.61 Å Release Date: 2022-08-17
Classification: HYDROLASE/HYDROLASE INHIBITOR
Ligands: GJN

6DF7 image
Taf1-Bd2 In Complex With Cpd27 (6-(But-3-En-1-Yl)-4-(1-Methyl-6-(Morpholine-4-Carbonyl)-1H-Benzo[D]Imidazol-4-Yl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)

6DF4 image
Taf1-Bd2 In Complex With Cpd8 (6-(But-3-En-1-Yl)-4-(3-(Morpholine-4-Carbonyl)Phenyl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)

5V84 image
Cecr2 In Complex With Cpd6 (6-Allyl-N,2-Dimethyl-7-Oxo-N-(1-(1-Phenylethyl)Piperidin-4-Yl)-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2017-06-14
Classification: Transcription/Inhibitor
Ligands: SO4, 96V

5LS6 image
Structure Of Human Polycomb Repressive Complex 2 (Prc2) With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.47 Å Release Date: 2017-02-22
Classification: Transferase/Inhibitor
Ligands: ZN, 74D

5I40 image
Brd9 In Complex With Cpd1 (6-Methyl-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.04 Å Release Date: 2016-10-12
Classification: RNA BINDING PROTEIN
Ligands: EDO, PEG, 67N

5I7X image
Brd9 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.18 Å Release Date: 2016-10-12
Classification: RNA BINDING PROTEIN
Ligands: 67B

5I7Y image
Brd9 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.45 Å Release Date: 2016-10-12
Classification: TRANSCRIPTION
Ligands: 69G

5I80 image
Brd4 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.45 Å Release Date: 2016-10-12
Classification: TRANSCRIPTION
Ligands: 67B, EDO, DMS

5I88 image
Brd4 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.40 Å Release Date: 2016-10-12
Classification: TRANSCRIPTION
Ligands: PGE, EDO, DMS, 69G, GOL

5I1Q image
Second Bromodomain Of Taf1 Bound To A Pyrrolopyridone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2016-06-08
Classification: PROTEIN BINDING/INHIBITOR
Ligands: 67C

5I29 image
Taf1(2) Bound To A Pyrrolopyridone Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.21 Å Release Date: 2016-06-08
Classification: PROTEIN BINDING/INHIBITOR
Ligands: 67B, CA

4JU3 image
Crystal Structure Of Hcv Ns5B Polymerase In Complex With Compound 8

4JU4 image
Crystal Structure Of Hcv Ns5B Polymerase In Complex With Compound 22

4JU6 image
Crystal Structure Of Hcv Ns5B Polymerase In Complex With Compound 24

4JU7 image
Crystal Structure Of Hcv Ns5B Polymerase In Complex With Compound 24
Protein Functional Filters:
Feedback Form
Name
Email
Institute
Feedback