Search Count: 16
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor Containing A Spiro-Bicyclic Group (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2021-08-11 Classification: HYDROLASE Ligands: ZN, SO4, CA, PEG, VJV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-08-11
Ligands: ZN, SO4, CA, PEG, VJV
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 20)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, SO4, PEG, WBA, DMS, WBD
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Structure Of Human Hdac2 In Complex With A 2-Substituted Benzamide Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2020-12-30 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, PEG, WB4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-30
Ligands: ZN, CA, PEG, WB4
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Structure Of Human Hdac2 In Complex With Ketone Inhibitor (Compound E)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2020-08-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, V1P |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: ZN, SO4, CA, PEG, V1P
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Structure Of Human Hdac2 In Complex With Ketone Inhibitor (Compound O)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2020-08-12 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, SO4, CA, PEG, V1S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: ZN, SO4, CA, PEG, V1S
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Structure Of Human Hdac2 In Complex With An Aryl Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2020-07-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, PEG, V1D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: ZN, CA, SO4, PEG, V1D
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Co-Structure Of Btk Kinase Domain With L-005085737 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULV, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULV, 5WE
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Co-Structure Of Btk Kinase Domain With L-005191930 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: ULY, 5WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: ULY, 5WE
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Co-Structure Of Btk Kinase Domain With L-005298385 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2020-07-22 Classification: TRANSFERASE Ligands: UM4, EDO, BTB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-22
Ligands: UM4, EDO, BTB
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: TV1, ZN, CA, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: TV1, ZN, CA, PEG
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Structure Of Human Hdac2 In Complex With An Ethyl Ketone Inhibitor Containing A Spiro-Bicyclic Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2020-05-06 Classification: HYDROLASE/HYDROLASE Inhibitor Ligands: ZN, SO4, CA, PEG, TV7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: ZN, SO4, CA, PEG, TV7
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Crystal Structure Of The Core Catalytic Domain Of Human O-Glcnacase Bound To Mk-8719
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2019-09-18 Classification: HYDROLASE Ligands: OQ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-09-18
Ligands: OQ1
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Thrombin In Complex With (S)-(4-Chloro-2-((1-(5-Methyl-1H-Pyrrole-2-Carbonyl)Pyrrolidine-2-Carboxamido)Methyl)Phenyl)Methanaminium
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2015-06-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: MG, GOL, NAG, 45S |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: MG, GOL, NAG, 45S
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Human Dipeptidyl Peptidase Iv/Cd26 In Complex With A 4-Aryl Cyclohexylalanine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: NAG, NA, 524 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: NAG, NA, 524
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Human Dipeptidyl Peptidase Iv/Cd26 In Complex With A 4-Aryl Cyclohexylalanine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2007-11-06 Classification: HYDROLASE Ligands: NAG, NA, 474 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-11-06
Ligands: NAG, NA, 474
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Human Dipeptidyl Peptidase Iv In Complex With An Alpha Amino Acid Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-05-08 Classification: HYDROLASE Ligands: NAG, NA, 277 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-05-08
Ligands: NAG, NA, 277
