Search Count: 13
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Human Tnf-Alpha In Complex With 2-[5-(3-Chloro-4-{[(1R)-1-(2-Fluorophenyl)Ethyl]Amino}Quinolin-6-Yl)Pyrimidin-2-Yl]Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2020-12-09 Classification: CYTOKINE Ligands: VGY, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-09
Ligands: VGY, GOL
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Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Novel Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2020-08-12 Classification: TRANSCRIPTION/Agonist Ligands: V27 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: V27
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Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Potent, Selective And Orally Bioavailable Ror-Gamma-T Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2020-08-12 Classification: TRANSCRIPTION/AGONIST Ligands: VBG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-12
Ligands: VBG, SO4
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244- 487)-L6-Src1(678-692)) In Complex With An Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-04-08 Classification: TRANSCRIPTION Ligands: R7V, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: R7V, GOL
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Structure Of Human Pregnane X Receptor Ligand Binding Domain Bound Tethered With Src Co-Activator Peptide And Compound-3 Aka 1,1,1,3,3,3-Hexafluoro-2-{4-[1-(4- Luorobenzenesulfonyl)Cyclopentyl]Phenyl}Propan-2-Ol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2020-02-12 Classification: TRANSFERASE Ligands: L7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-12
Ligands: L7D
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis- Rorgt(244-487)-L6-Src1(678-692)) In Complex With A Tricyclic Inverse Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2019-11-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: O5B, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: O5B, GOL
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With A Phenyl (3-Phenylpyrrolidin-3-Yl)Sulfone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-07-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: O5A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: O5A
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Crystal Structure Of Rar-Related Orphan Receptor C In Complex With A Phenyl (3-Phenylpyrrolidin-3-Yl)Sulfone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2019-03-20 Classification: TRANSCRIPTION/INHIBITOR Ligands: L8A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-20
Ligands: L8A
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Identification Of Bicyclic Hexafluoroisopropyl Alcohol Sulfonamides As Rorgt/Rorc Inverse Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-12-20 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: XGH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: XGH, SO4
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Structure Of Human Pregnane X Receptor Ligand Binding Domain Bound Tethered With Src Co-Activator Peptide And Compound 25A Aka Bicyclic Hexafluoroisopropyl 2 Alcohol Sulfonamides
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.56 Å Release Date: 2017-12-20 Classification: NUCLEAR PROTEIN Ligands: XGH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: XGH
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The Jak3 Kinase Domain In Complex With A Covalent Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.48 Å Release Date: 2017-10-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 9Z4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-10-04
Ligands: 9Z4
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-05-31 Classification: TRANSFERASE/INHIBITOR Ligands: 9J4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-05-31
Ligands: 9J4
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Crystal Structure Of Jak3 Kinase Domain In Complex With A Pyrrolopyridazine Carboxamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2014-12-24 Classification: TRANSFERASE/INHIBITOR Ligands: 3QX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3QX