Search Count: 7
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Fragment-Based Discovery Of Focal Adhesion Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2013-09-11 Classification: Transferase/Transferase Inhibitor Ligands: K8A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: K8A
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Focal Adhesion Kinase Catalytic Domain In Complex With 1-[4-(6-Amino-Purin-9-Yl)-Phenyl]-3-(5-Tert-Butyl-2-P-Tolyl-2H-Pyrazol-3-Yl)-Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2013-09-11 Classification: Transferase/Transferase Inhibitor Ligands: K9Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: K9Y
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Focal Adhesion Kinase Catalytic Domain In Complex With 3-Methyl-1,4-Dihydro-Pyrazolo[4,5-C]Pyrazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2013-09-11 Classification: Transferase/Transferase Inhibitor Ligands: 4KA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: 4KA
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Focal Adhesion Kinase Catalytic Domain In Complex With 1-(5-Tert-Butyl-2-P-Tolyl-2H-Pyrazol-3-Yl)-3-(4-Pyridin-3- Yl-Phenyl)-Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2013-09-11 Classification: Transferase/Transferase Inhibitor Ligands: KAO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-11
Ligands: KAO, SO4
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Structural And Biophysical Characterization Of The Syk Activation Switch
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2012-11-28 Classification: TRANSFERASE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: ANP, MG
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Structural And Biophysical Characterization Of The Syk Activation Switch
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2012-11-28 Classification: TRANSFERASE Ligands: MG, ANP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: MG, ANP
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Structural And Biophysical Characterization Of The Syk Activation Switch
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-11-28 Classification: TRANSFERASE Ligands: ANP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-28
Ligands: ANP, MG
