Search Count: 29
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Human Spleen Tyrosine Kinase Kinase Domain In Complex With Azanaphthyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2016-09-14 Classification: TRANSFERASE Ligands: 6ZG, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: 6ZG, GOL, DMS
 |
Human Spleen Tyrosine Kinase Kinase Domain In Complex With Azanaphthyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-09-14 Classification: TRANSFERASE Ligands: 6ZF, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: 6ZF, GOL
 |
Crystal Structure Of Human Atad2 Bromodomain In Complex With 8-(((3R,4R,5S)-3-((4,4-Difluorocyclohexyl)Methoxy)-5-Methoxypiperidin-4-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XX, SO4
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N-Terminal Bromodomain Of Human Brd4 With 8-(((3R,4R,5S)-3-((4,4-Difluorocyclohexyl)Methoxy)-5-Methoxypiperidin-4-Yl)Amino)-3-Methyl-5-(5-Methylpyridin-3-Yl)-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XX
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N-Terminal Bromodomain Of Human Brd4 With 5-(5-Aminopyridin-3-Yl)-8-(((3R,4R)-3-((1,1-Dioxidotetrahydro-2H-Thiopyran-4-Yl)Methoxy)Piperidin-4-Yl)Amino)-3-Methyl-1,7-Naphthyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2016-08-31 Classification: TRANSCRIPTION Ligands: EDO, 6XW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-08-31
Ligands: EDO, 6XW
 |
Cell Penetrant Inhibitors Of The Jmjd2 (Kdm4) And Jarid1 (Kdm5) Families Of Histone Lysine Demethylases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: YC8, ZN, MG, BCN, CO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: YC8, ZN, MG, BCN, CO
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Crystal Structure Of Human Kdm4D In Complex With 3-(4- Phenylbutanamido)Pyridine-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-01-27 Classification: TRANSCRIPTION Ligands: ZN, FE2, GOL, YC8, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, FE2, GOL, YC8, SO4
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Crystal Structure Of Human Kdm4D In Complex With 3-4-Methylthiophen-2- Ylmethylaminopyridine-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: ZN, CO, AUY, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, CO, AUY, SO4
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Crystal Structure Of Human Kdm4D In Complex With 3-Aminopyridine-4- Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: ZN, CO, GOL, 4SV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, CO, GOL, 4SV, SO4
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Crystal Structure Of Human Kdm4D In Complex With 3H,4H-Pyrido-3,4-D- Pyrimidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: ZN, CO, N5J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, CO, N5J, SO4
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Crystal Structure Of Human Kdm4D In Complex With 2-1H-Pyrazol-4-Yloxy- 3H,4H-Pyrido-3,4-D-Pyrimidin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2016-01-27 Classification: OXIDOREDUCTASE Ligands: ZN, CO, HA6, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-27
Ligands: ZN, CO, HA6, SO4
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000222
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DF, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DF, GOL
 |
The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000223
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DL, DMS
 |
Syk Kinase Domain In Complex With Inhibitor Gtc000224
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DK
 |
Syk Kinase Domain In Complex With Inhibitor Gtc000225
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DJ
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000226
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DN
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000233
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: GOL, 4DQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: GOL, 4DQ
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000249
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DO
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 8-(3R,4R) -3-(Cyclohexylmethoxy)Piperidin-4-Yl-Amino-3-Methyl-1,2-Dihydro-1,7- Naphthyridin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-08-12 Classification: HYDROLASE Ligands: EDO, 78J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: EDO, 78J, SO4
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Crystal Structure Of Human Atad2 Bromodomain In Complex With 4-(3R,4R) -4-(3-Methyl-2-Oxo-1,2-Dihydro-1,7-Naphthyridin-8-Yl)Aminopiperidin-3- Yloxymethyl)-1-Thiane-1,1-Dione
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2015-08-12 Classification: INHIBITOR Ligands: EDO, YEJ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-12
Ligands: EDO, YEJ, SO4