Search Count: 13
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Identification Of M4205 A Highly Selective Inhibitor Of Ckit Mutations For Unresectable Metastatic Or Recurrent Gist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2023-02-22 Classification: TRANSFERASE Ligands: K3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: K3R
 |
Identification Of M4205 A Highly Selective Inhibitor Of Ckit Mutations For Unresectable Metastatic Or Recurrent Gist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.09 Å Release Date: 2023-02-22 Classification: TRANSFERASE Ligands: KCI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-22
Ligands: KCI
 |
Human Tnks1 In Complex With 3-[4-(1-Hydroxy-1-Methyl-Ethyl)-Phenyl]-6-Methyl-2H-Pyrrolo[1,2-A]Pyrazin-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2021-07-28 Classification: TRANSFERASE Ligands: ACT, V8B, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: ACT, V8B, ZN
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Human Tnks1 In Complex With 6,8-Difluoro-2-[4-(1-Hydroxy-1-Methyl-Ethyl)-Phenyl]-3H-Quinazolin-4-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2019-08-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BME, JKN, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-14
Ligands: BME, JKN, ZN
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Discovery Of Novel 7-Azaindoles As Pdk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: SO4, 61Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: SO4, 61Y
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Discovery Of Novel 7-Azaindoles As Pdk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: SO4, 62O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: SO4, 62O
 |
Discovery Of Novel 7-Azaindoles As Pdk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: 63L, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 63L, SO4
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Discovery Of Novel 7-Azaindoles As Pdk1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2016-06-08 Classification: TRANSFERASE Ligands: 63E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-08
Ligands: 63E, SO4
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Identification And Optimization Of Pyridazinones As Potent And Selective C-Met Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2015-03-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3E8, GBL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3E8, GBL
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Identification And Optimization Of Pyridazinones As Potent And Selective C-Met Kinase Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-03-18 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3EH, 7PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-18
Ligands: 3EH, 7PE
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Rapid Preparation Of Triazolyl Substituted Nh-Heterocyclic Kinase Inhibitors Via One-Pot Sonogashira Coupling Tms-Deprotection Cuaac Sequence
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2011-06-15 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3RC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-06-15
Ligands: 3RC
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Factor Xa Specific Inhibitor In Complex With Bovine Trypsin
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2000-08-25 Classification: SERINE PROTEASE Ligands: CA, SO4, ZEN |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2000-08-25
Ligands: CA, SO4, ZEN
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Factor Xa Specific Inhibitor In Complex With Bovine Trypsin
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2000-08-25 Classification: SERINE PROTEASE Ligands: CA, SO4, ZEN |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2000-08-25
Ligands: CA, SO4, ZEN