Search Count: 21
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Crystal Structure Of Human Il-17A In Complex With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2025-10-15 Classification: CYTOKINE Ligands: A1CXF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-15
Ligands: A1CXF
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Il17A Homodimer Complexed To Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCE
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Il17A Complexed To Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2024-04-03 Classification: CYTOKINE Ligands: XCW, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-04-03
Ligands: XCW, CL
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Crystal Structure Of Setdb1 Tudor Domain In Complex With Mr46747
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2023-11-22 Classification: TRANSFERASE Ligands: XRU, SO4, EDO, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: XRU, SO4, EDO, UNX
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Crystal Structure Of Wild-Type C-Met Bound By Compound 7.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2022-08-31 Classification: TRANSFERASE Ligands: SO4, MDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: SO4, MDI
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Crystal Structure Of D1228V C-Met Bound By Compound 1.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2022-08-31 Classification: TRANSFERASE Ligands: GOL, MDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-31
Ligands: GOL, MDI
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Crystal Structure Of The Wdr Domain Of Human Dcaf1 In Complex With Oicr-6766
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-05-04 Classification: TRANSFERASE Ligands: N6O, UNX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-04
Ligands: N6O, UNX
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Mertk Kinase Domain In Complex With Nps-1034
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4K
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Mertk Kinase Domain In Complex With Quinazoline-Based Inhbitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4E, SO4
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Mertk Kinase Domain In Complex With A Bisaminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4N
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Mertk Kinase Domain In Complex With Purine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Q
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Mertk Kinase Domain In Complex With A Type 2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4T
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Mertk Kinase Domain With Type 1.5 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4W
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Mertk Kinase Domain With Type 1 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Z
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Mertk Kinase Domain With Type 3 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S5E, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S5E, CL, EDO
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Sirt1/Activator Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-07-15 Classification: Hydrolase/hydrolase activator Ligands: ZN, 4TO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-15
Ligands: ZN, 4TO
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Sirt1/Activator/Inhibitor Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2015-07-15 Classification: Hydrolase/hydrolase inhibitor Ligands: 4TQ, 1NS, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-15
Ligands: 4TQ, 1NS, ZN
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Sirt1/Activator/Substrate Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2015-07-15 Classification: HYDROLASE Ligands: ZN, CNA, 4TQ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-15
Ligands: ZN, CNA, 4TQ, GOL
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Crystal Structure Of Human Sirt3 With Elt Inhibitor 11C [N-{2-[1-(6-Carbamoylthieno[3,2-D]Pyrimidin-4-Yl)Piperidin-4-Yl]Ethyl}-N'-Ethylthiophene-2,5-Dicarboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-04-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 1NQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: ZN, 1NQ
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Crystal Structure Of Human Sirt3 With Elt Inhibitor 28 [4-(4-{2-[(2,2-Dimethylpropanoyl)Amino]Ethyl}Piperidin-1-Yl)Thieno[3,2-D]Pyrimidine-6-Carboxamide[
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2013-04-24 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 1NR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-04-24
Ligands: ZN, 1NR
