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9MNR image
Panoptes Opts Minimal Crispr Polymerase (Mcpol) From Klebsiella Pneumoniae Strain Kp67

9PD0 image
Panoptes Opts Minimal Crispr Polymerase (Mcpol) With Non-Hydrolyzable Ligand Apcpp From Klebsiella Pneumoniae Strain Kp67

7SUB image
3-Oxoacyl-Acp Reductase Fabg

6EEY image
Crystal Structure Of Human Scribble Pdz4 R1110G Mutant

4W2R image
Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-2-[(4-Methoxy-6-Methyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-7-[(R)-Methoxy(Oxetan-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One

6B3W image
Structure Of Hs/Acprc2 In Complex With 5,8-Dichloro-7-(3,5-Dimethyl-1,2-Oxazol-4-Yl)-2-[(4,6-Dimethyl-2-Oxo-1,2-Dihydropyridin-3-Yl)Methyl]-3,4-Dihydroisoquinolin-1(2H)-One

5UG8 image
Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With A Covalent Inhibitor N-[(3R,4R)-4-Fluoro-1-{6-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-9-(Propan-2-Yl)-9H-Purin-2-Yl}Pyrrolidin-3-Yl]Propanamide

5UG9 image
Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With A Covalent Inhibitor N-[(3R,4R)-4-Fluoro-1-{6-[(3-Methoxy-1-Methyl-1H-Pyrazol-4-Yl)Amino]-9-(Propan-2-Yl)-9H-Purin-2-Yl}Pyrrolidin-3-Yl]Propanamide

5UGA image
Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With 4-(4-{[2-{[(3S)-1-Acetylpyrrolidin-3-Yl]Amino}-9-(Propan-2-Yl)-9H-Purin-6-Yl]Amino}Phenyl)-1-Methylpiperazin-1-Ium

5UGB image
Crystal Structure Of The Egfr Kinase Domain In Complex With 4-(4-{[2-{[(3S)-1-Acetylpyrrolidin-3-Yl]Amino}-9-(Propan-2-Yl)-9H-Purin-6-Yl]Amino}Phenyl)-1-Methylpiperazin-1-Ium

5UGC image
Crystal Structure Of The Egfr Kinase Domain (L858R, T790M, V948R) In Complex With A Covalent Inhibitor N-[(3R,4R)-4-Fluoro-1-{6-[(3-Methoxy-1-Methyl-1H-Pyrazol-4-Yl)Amino]-9-Methyl-9H-Purin-2-Yl}Pyrrolidin-3-Yl]Propanamide

5KZ0 image
Structure Of Human Anaplastic Lymphoma Kinase In Complex With 2-[(1R)-1-{[2-Amino-5-(1,3-Dimethyl-1H-Pyrazol-4-Yl)Pyridin-3-Yl]Oxy}Ethyl]-4-Fluoro-N,N-Dimethylbenzamide

5HG5 image
Egfr (L858R, T790M, V948R) In Complex With N-{3-[(2-{[4-(4-Methylpiperazin-1-Yl)Phenyl]Amino}-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl)Oxy]Phenyl}Prop-2-Enamide

5HG8 image
Egfr (L858R, T790M, V948R) In Complex With N-[3-({2-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl}Oxy)Phenyl]Prop-2-Enamide

5HG9 image
Egfr (L858R, T790M, V948R) In Complex With 1-[(3R,4R)-3-[({2-[(1-Methyl-1H-Pyrazol-4-Yl)Amino]-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yl}Oxy)Methyl]-4-(Trifluoromethyl)Pyrrolidin-1-Yl]Prop-2-En-1-One

5HG7 image
Egfr (L858R, T790M, V948R) In Complex With 1-{(3R,4R)-3-[5-Chloro-2-(1-Methyl-1H-Pyrazol-4-Ylamino)-7H-Pyrrolo[2,3-D]Pyrimidin-4-Yloxymethyl]-4-Methoxy-Pyrrolidin-1-Yl}Propenone (Pf-06459988)

4CLI image
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With Pf- 06463922 ((10R)-7-Amino-12-Fluoro-2,10,16-Trimethyl-15-Oxo-10,15,16, 17-Tetrahydro-2H-8,4-(Metheno)Pyrazolo(4,3-H)(2,5,11) Benzoxadiazacyclotetradecine-3-Carbonitrile).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2014-05-28
Classification: TRANSFERASE
Ligands: 5P8

4CLJ image
Structure Of L1196M Mutant Human Anaplastic Lymphoma Kinase In Complex With Pf-06463922 ((10R)-7-Amino-12-Fluoro-2,10,16-Trimethyl- 15-Oxo-10,15,16,17-Tetrahydro-2H-8,4-(Metheno)Pyrazolo(4,3-H)(2,5,11) Benzoxadiazacyclotetradecine-3-Carbonitrile).
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.66 Å Release Date: 2014-05-28
Classification: TRANSFERASE
Ligands: 5P8

4CMO image
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With The Inhibitor 2-((1R)-1-((3-Amino-6-(2-Methoxypyridin-3-Yl)Pyrazin-2-Yl) Oxy)Ethyl)-4-Fluoro-N-Methylbenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2014-05-28
Classification: TRANSFERASE
Ligands: YPW

4CMT image
Structure Of The Human Anaplastic Lymphoma Kinase In Complex With The Inhibitor 3-((1R)-1-(5-Fluoro-2-(2H-1,2,3-Triazol-2-Yl)Phenyl)Ethoxy)- 5-(3-(Methylsulfonyl)Phenyl)Pyridin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.73 Å Release Date: 2014-05-28
Classification: TRANSFERASE
Ligands: GWH
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