Search Count: 10
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Tead1/Yap In Complex With A Reversible Inhibitor N-[(4-Phenoxyphenyl)Methyl]Imidazo[1,2-A]Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2024-10-16 Classification: TRANSCRIPTION Ligands: CL, A1IHH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-16
Ligands: CL, A1IHH
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Optimization Of Tead P-Site Binding Fragment Hit Into In Vivo Active Lead Msc-4106
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JJU, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JJU, SO4
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Human Tead3 In Complex With 1-Cyclopentyl-1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JIK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JIK
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Prmt5:Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
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Prmt5:Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2021-11-17 Classification: Transferase/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
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Prmt5:Mep50 Complexed With Adenosine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ADN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ADN
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06855800
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2021-11-17 Classification: TRANSFERASE/Transcription Ligands: ZR4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR4
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Prmt5(M420T Mutant):Mep50 Complexed With Inhibitor Pf-06939999
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2021-11-17 Classification: transferase/Transcription Ligands: ZR1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-17
Ligands: ZR1
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Structure Of Sasanlimab Fab In Complex With Pd-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2020-09-09 Classification: ANTITUMOR PROTEIN/IMMUNE SYSTEM Ligands: GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-09
Ligands: GOL
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A Novel Small Molecule Apkc Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2013-02-27 Classification: TRANSFERASE Ligands: IOD, CL, C58, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-02-27
Ligands: IOD, CL, C58, EDO
