Search Count: 5
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Jak1 Kinase (Jh1 Domain) In Complex With Povorcitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2026-06-10 Classification: TRANSFERASE Ligands: EDO, A1C68, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: EDO, A1C68, DMS
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Jak2 Kinase (Jh1 Domain) In Complex With Povorcitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2026-06-10 Classification: TRANSFERASE Ligands: MLA, A1C68 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-10
Ligands: MLA, A1C68
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Discovery Of An Orally Biovailable Kras G12D Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2025-01-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GDP, MG, A1BEI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: GDP, MG, A1BEI
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Discovery Of An Orally Bioavailable Kras G12D Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-01-22 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GDP, A1BEJ, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-22
Ligands: GDP, A1BEJ, MG
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Discovery Of (4-Pyrazolyl)-2-Aminopyrimidines As Potent And Selective Inhibitors Of Cyclin-Dependent Kinase 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2024-02-14 Classification: TRANSFERASE/INHIBITOR Ligands: XKU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: XKU
