Search Count: 16
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Human Pi3K P85Alpha/P110Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
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P85Alpha/P110Alpha Heterodimer H1047R Mutant
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.72 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
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Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UE9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UE9
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Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UIW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UIW
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Human Pi3K P85Alpha/P110Alpha Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.53 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UIW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UIW
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Human Pi3K P85Alpha/P110Alpha H1047R Bound To Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.62 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN/INHIBITOR Ligands: UJC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: UJC
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Human Pi3K P85Alpha/P110Alpha Bound To Rly-2608
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2023-11-22 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: XUZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-11-22
Ligands: XUZ
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Cryoem Structure Of Pi3Kalpha
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-11-15 Classification: CYTOSOLIC PROTEIN |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-11-15
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Tankyrase-1 Complexed With Small Molecule Inhibitor N-[(4-Oxo-3,4-Dihydroquinazolin-2-Yl)Methyl]-3-Phenyl-N-(Thiophen-2-Ylmethyl)Propanamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-08-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, SO4, 1XO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: ZN, SO4, 1XO
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Tankyrase-1 Complexed With Small Molecule Inhibitor 4-Chloro-5-Cyano-N-{2-[4-(4-Fluorobenzoyl)Piperidin-1-Yl]Ethyl}-2-Methoxybenzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-08-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, NA, 1XP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: SO4, NA, 1XP
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Tankyrase-1 Complexed With Small Molecule Inhibitor 2-[4-(4-Fluorobenzoyl)Piperidin-1-Yl]-N-[(4-Oxo-3,5,7,8-Tetrahydro-4H-Pyrano[4,3-D]Pyrimidin-2-Yl)Methyl]-N-(Thiophen-2-Ylmethyl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2013-08-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: ZN, 1XQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-14
Ligands: ZN, 1XQ, SO4
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Crystal Structure Of Human Bcl-2 In Complex With A Small Molecule Inhibitor Targeting Bcl-2 Bh3 Domain Interactions
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-07-10 Classification: APOPTOSIS/INHIBITOR Ligands: 1E9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-10
Ligands: 1E9
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Benzamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2008-04-08 Classification: TRANSFERASE Ligands: RAJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-08
Ligands: RAJ
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Naphthamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2008-04-01 Classification: TRANSFERASE Ligands: 900 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-04-01
Ligands: 900
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Benzimidazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: 276 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: 276
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With A Benzoxazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2007-09-25 Classification: TRANSFERASE Ligands: SO4, 857 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-25
Ligands: SO4, 857
