Search Count: 27
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Crystal Structure Of The Complex Between Vhl, Elonginb, Elonginc, And Compound 5
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2024-05-29 Classification: TRANSCRIPTION Ligands: TFA, PEG, EDO, ACT, DMS |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: TFA, PEG, EDO, ACT, DMS
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Crystal Structure Of The Complex Between Vhl, Elonginb, Elonginc, And Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2024-05-29 Classification: TRANSCRIPTION Ligands: EDO, DMS, CL, A1ARP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, DMS, CL, A1ARP
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Gdc-9545 In Complex With Estrogen Receptor Alpha
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2021-06-02 Classification: TRANSCRIPTION Ligands: G9J, ZNM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-02
Ligands: G9J, ZNM
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Crystal Structure Of Braf In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: V5J, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: V5J, IOD
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Crystal Structure Of Braf In Complex With Inhibitor Gne-0749
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VQP, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: VQP, CL
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Crystal Structure Of Htdo2 Bound To Inhibitor Gne1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.18 Å Release Date: 2020-05-06 Classification: OXIDOREDUCTASE/Inhibitor Ligands: HEM, QVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-06
Ligands: HEM, QVY
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Ldha Structure In Complex With Inhibitor 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2019-10-30 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAI, EPE, SO4, D3S, LAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-30
Ligands: NAI, EPE, SO4, D3S, LAC
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Ldha Structure In Complex With Inhibitor 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2019-10-30 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NAI, EPE, SO4, D4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-30
Ligands: NAI, EPE, SO4, D4S
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Crystal Structure Of Irak4 In Complex With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-05-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: LS7, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: LS7, SO4, GOL
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Structure Of The Irak4 Kinase Domain With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: CA, LRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: CA, LRS
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Structure Of The Irak4 Kinase Domain With Compound 41
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: SO4, LSV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: SO4, LSV
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Structure Of The Irak4 Kinase Domain With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2019-05-22 Classification: IMMUNE SYSTEM Ligands: LTY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-22
Ligands: LTY
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Lactate Dehydrogenase In Complex With Inhibitor 6-(3-Aminophenyl)-3-((2-Chlorophenyl)Thio)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, EPE, SO4, D4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, EPE, SO4, D4S
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Lactate Dehydrogenase In Complex With Inhibitor (S)-5-((2-Chlorophenyl)Thio)-6'-((4-Fluorophenyl)Amino)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: EPE, NAD, LAC, SO4, D47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: EPE, NAD, LAC, SO4, D47
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Lactate Dehydrogenase In Complex With Inhibitor (R)-3-((2-Chlorophenyl)Thio)-6-(3-((4-Fluorophenyl)Amino)Phenyl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE Ligands: NAD, EPE, SO4, D3S, LAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, EPE, SO4, D3S, LAC
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Lactate Dehydrogenase In Complex With Inhibitor (R)-5-((2-Chlorophenyl)Thio)-6'-(4-Fluorophenoxy)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, D3J, LAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, D3J, LAC
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Lactate Dehydrogenase In Complex With Inhibitor (S)-5-((2-Chlorophenyl)Thio)-6'-(4-Fluorophenoxy)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, LAC, D4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, LAC, D4J
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Lactate Dehydrogenase In Complex With Inhibitor 3-((2-Chlorophenyl)Thio)-6-(6-((4-Fluorophenyl)Amino)Pyridin-2-Yl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, D4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, D4A
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Lactate Dehydrogenase In Complex With Inhibitor (R)-3-((2-Chlorophenyl)Thio)-6-(3-((4-Fluorophenyl)Amino)Phenyl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-10-17 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, EPE, SO4, D0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: NAD, EPE, SO4, D0Y
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Lactate Dehydrogenase In Complex With Inhibitor (R)-5-((2-Chlorophenyl)Thio)-6'-((4-Fluorophenyl)Amino)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-10-17 Classification: OXIDOREDUCTASE/Inhibitor Ligands: EPE, NAD, SO4, D0V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: EPE, NAD, SO4, D0V
