Search Count: 22
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Structure Of Sos1 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2025-09-17 Classification: CYTOSOLIC PROTEIN Ligands: A1I6H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-17
Ligands: A1I6H
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Fragment Screening Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2025-06-18 Classification: GENE REGULATION Ligands: A1I5P, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
Ligands: A1I5P, ZN
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Tricyclic Pyrimidoindolone Inhibitor (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-05-14 Classification: GENE REGULATION Ligands: A1I45, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1I45, ZN
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd5305 (Saruparib)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H63, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H63, SO4
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Crystal Structure Of Parp1 Catalytic Domain Bound To Azd9574
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2024-12-04 Classification: TRANSFERASE Ligands: A1H64, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-04
Ligands: A1H64, SO4
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Crystal Structure Of Mus81-Eme1, Apo Form.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2024-07-03 Classification: HYDROLASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
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Crystal Structure Of Mus81-Eme1 Bound By Compound 15.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2024-07-03 Classification: HYDROLASE Ligands: MG, A1IA7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, A1IA7
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Crystal Structure Of Mus81-Eme1 Bound By Compound 16.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2024-07-03 Classification: HYDROLASE Ligands: MG, EOH, A1IA8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-07-03
Ligands: MG, EOH, A1IA8
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Crystal Structure Of Mus81-Eme1 Bound By Compound 10.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2024-06-19 Classification: HYDROLASE Ligands: A1IA5, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-19
Ligands: A1IA5, MG
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Crystal Structure Of Mus81-Eme1 Bound By Compound 12.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.91 Å Release Date: 2024-06-19 Classification: HYDROLASE Ligands: A1IA6, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-19
Ligands: A1IA6, MG
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Crystal Structure Of Mus81-Eme1 Bound By Compound 21.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2024-06-19 Classification: HYDROLASE Ligands: MG, A1IA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-19
Ligands: MG, A1IA4
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Crystal Structure Of The Pwwp1 Domain Of Nsd2 Bound By Compound 17.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.43 Å Release Date: 2024-05-29 Classification: TRANSFERASE Ligands: EDO, A1H7X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, A1H7X
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Crystal Structure Of The Pwwp1 Domain Of Nsd2 Bound By Compound 18.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2024-05-29 Classification: TRANSFERASE Ligands: EDO, EOH, A1H7Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: EDO, EOH, A1H7Y
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Crystal Structure Of The Pwwp1 Domain Of Nsd2 Bound By Compound 34.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-05-29 Classification: TRANSFERASE Ligands: A1H7Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-29
Ligands: A1H7Z
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Parp1 Catalytic Domain In Complex With 8-Chloroquinazolinone-Based Inhibitor (Compound 9)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKW, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKW, SO4
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Parp1 Catalytic Domain In Complex With Isoquinolone-Based Inhibitor (Compound 16)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKT, SO4
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Parp1 Catalytic Domain In Complex With A Selective Pyridine Carboxamide-Based Inhibitor (Compound 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VKQ, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VKQ, SO4
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Mek1 In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-03-03 Classification: TRANSFERASE Ligands: MG, ANP, SU5, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: MG, ANP, SU5, SO4
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Mek1 In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2021-03-03 Classification: TRANSFERASE Ligands: ANP, MG, T1K, SO4, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: ANP, MG, T1K, SO4, PO4
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Mek1 In Complex With Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-03-03 Classification: TRANSFERASE Ligands: ANP, MG, T3W, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: ANP, MG, T3W, SO4
