Search Count: 7
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To Amg 510
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-11-06 Classification: SIGNALING PROTEIN Ligands: MG, GDP, MOV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: MG, GDP, MOV
![]() |
Discovery Of Mk-8353: An Orally Bioavailable Dual Mechanism Erk Inhibitor For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-08-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, G67 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-08-08
Ligands: SO4, G67
![]() |
Discovery Of 3(S)-Thiomethyl Pyrrolidine Erk Inhibitors For Oncology
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: SO4, F8V |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: SO4, F8V
![]() |
Crystal Structure Of Heptaprenyl Diphosphate Synthase From Staphylococcus Aureus
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2016-12-28 Classification: TRANSFERASE Ligands: PO4 |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2016-12-28
Ligands: PO4
![]() |
Crystal Structure Of The Ternary Human Pl Kinase-Ginkgotoxin-Mgatp Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2012-05-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, NA, ATP, GT0, MPD, SO4, GT1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-02
Ligands: MG, NA, ATP, GT0, MPD, SO4, GT1
![]() |
Crystal Structure Of Human Pl Kinase With Bound Theophylline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2012-05-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-05-02
![]() |
Discovery Of C-Imidazole Azaheptapyridine Fpt Inhibitors
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-01-26 Classification: TRANSFERASE Ligands: MG, ZN, FPP, Z96 |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2010-01-26
Ligands: MG, ZN, FPP, Z96
