Search Count: 25
![]() |
Krasg12C Gdp Form In Complex With Cpd3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2021-10-13 Classification: ONCOPROTEIN Ligands: GDP, MG, PO4, QWK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: GDP, MG, PO4, QWK
![]() |
Krasg12C Gdp Form In Complex With Cpd1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2021-10-13 Classification: ONCOPROTEIN Ligands: GDP, MG, QWB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: GDP, MG, QWB
![]() |
Krasg12C Gdp Form In Complex With Cpd2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-10-13 Classification: ONCOPROTEIN Ligands: QWH, GDP, MG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: QWH, GDP, MG, SO4
![]() |
Krasg12C Gdp Form In Complex With Cpd4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2021-10-13 Classification: ONCOPROTEIN Ligands: GDP, QY5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-10-13
Ligands: GDP, QY5
![]() |
Sar156497 An Exquisitely Selective Inhibitor Of Aurora Kinases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-11-19 Classification: TRANSFERASE Ligands: Y3M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: Y3M
![]() |
Sar156497 An Exquisitely Selective Inhibitor Of Aurora Kinases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2014-11-19 Classification: TRANSFERASE Ligands: QMN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: QMN
![]() |
Sar156497 An Exquisitely Selective Inhibitor Of Aurora Kinases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-11-19 Classification: TRANSFERASE Ligands: JVE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: JVE
![]() |
Discovery And Optimization Of Pyrimidone Indoline Amide Pi3Kbeta Inhibitors For The Treatment Of Phosphatase And Tensin Homologue (Pten)-Deficient Cancers
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-01-15 Classification: TRANSFERASE Ligands: J82 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-01-15
Ligands: J82
![]() |
Crystal Structure Of Mek1 In Complex With Fragment 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-05-22 Classification: TRANSFERASE Ligands: 92P, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 92P, NA
![]() |
Crystal Structure Of Mek1 In Complex With Fragment 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2013-05-22 Classification: TRANSFERASE Ligands: MT8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: MT8
![]() |
Crystal Structure Of Mek1 In Complex With Fragment 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-05-22 Classification: TRANSFERASE Ligands: 5EZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 5EZ
![]() |
Crystal Structure Of Mek1 In Complex With Fragment 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2013-05-22 Classification: TRANSFERASE Ligands: YSO, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: YSO, NA
![]() |
Crystal Structure Of Mek1 In Complex With Fragment 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2013-05-22 Classification: TRANSFERASE Ligands: 22T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-05-22
Ligands: 22T
![]() |
X-Ray Structure Of Pi3K-Gamma Bound To A 4-(Morpholin-4-Yl)- (6-Oxo-1,6-Dihydropyrimidin-2-Yl)Amide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2012-11-14 Classification: Transferase/Transferase Inhibitor Ligands: 0W7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 0W7
![]() |
Structure Of Candida Albicans Kar3 Motor Domain Fused To Maltose-Binding Protein
Organism: Escherichia coli, Candida albicans
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2012-10-10 Classification: MOTOR PROTEIN Ligands: MG, ADP, EDO |
Organism: Escherichia coli, Candida albicans
Method: X-RAY DIFFRACTION
Release Date: 2012-10-10
Ligands: MG, ADP, EDO
![]() |
Discovery And Optimization Of New Benzimidazole- And Benzoxazole-Pyrimidone Selective Pi3Kbeta Inhibitors For The Treatment Of Phosphatase And Tensin Homologue (Pten)-Deficient Cancers
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-05-16 Classification: TRANSFERASE Ligands: VWN |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2012-05-16
Ligands: VWN
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2011-10-26 Classification: CHAPERONE Ligands: YK9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-26
Ligands: YK9
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJW
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJX
![]() |
Tricyclic Series Of Hsp90 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2011-10-19 Classification: CHAPERONE Ligands: YJW, YJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-10-19
Ligands: YJW, YJX
