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10KT image
Crystal Structure Of A2A Adenosine Receptor A2Ar-Bril In Complex With Compound50
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Resolution:2.59 Å Release Date: 2026-05-20
Classification: MEMBRANE PROTEIN

8E80 image
Structure Of Lrrk2-Chk1 10-Pt. Mutant Complex With Heteroaryl-1H-Indazole Lrrk2 Inhibitor 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.49 Å Release Date: 2023-02-22
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: UUF

8E81 image
Structure Of Lrrk2-Chk1 10-Pt. Mutant Complex With Heteroaryl-1H-Indazole Lrrk2 Inhibitor 25
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.62 Å Release Date: 2023-02-22
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: UU6

5U6I image
Discovery Of Mli-2, An Orally Available And Selective Lrrk2 Inhibitor That Reduces Brain Kinase Activity
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Resolution:1.69 Å Release Date: 2017-03-15
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: 81Y, SO4
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