Search Count: 21
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C-Terminal Bromodomain Of Human Brd2 With 5-(1-Benzyl-4-Chloro-1H-Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2024-06-26 Classification: TRANSCRIPTION Ligands: EDO, PE4, A1IBV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: EDO, PE4, A1IBV
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N-Terminal Bromodomain Of Human Brd4 With (5-(4-Chloro-1-((Tetrahydro-2H-Pyran-4-Yl)Methyl)-1H-Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-06-26 Classification: TRANSCRIPTION Ligands: EDO, A1IB5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-06-26
Ligands: EDO, A1IB5
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N-Terminal Bromodomain Of Human Brd2 With 5-(4-(4-Fluorophenyl)-1H-Imidazol-5-Yl)-1-Methylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-02-19 Classification: TRANSCRIPTION Ligands: SO4, NUQ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-02-19
Ligands: SO4, NUQ, EDO
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N-Terminal Bromodomain Of Human Brd4 With 1-((1-Acetylpiperidin-4-Yl)Methyl)-2-(4-Hydroxy-3,5-Dimethylphenyl)-N-Methyl-1H-Benzo[D]Imidazole-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: NUW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: NUW, EDO
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N-Terminal Bromodomain Of Human Brd4 With 1,3-Dimethyl-5-(1-((Tetrahydro-2H-Pyran-4-Yl)Methyl)-1H-Benzo[D]Imidazol-2-Yl)Pyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: EDO, NUB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: EDO, NUB
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N-Terminal Bromodomain Of Human Brd4 With 5-(1-(1,3-Dimethoxypropan-2-Yl)-5-Morpholino-1H-Benzo[D]Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: EDO, NV2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: EDO, NV2
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N-Terminal Bromodomain Of Human Brd4 With 5-(1-(1,3-Dimethoxypropan-2-Yl)-5-Morpholino-1H-Benzo[D]Imidazol-2-Yl)-1,3-Dimethylpyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2020-01-15 Classification: TRANSCRIPTION Ligands: SO4, NUH, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-01-15
Ligands: SO4, NUH, EDO
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Crystal Structure Of Spleen Tyrosine Kinase (Syk) In Complex With A 2-(Pyridinyloxymethyl)Pyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-10-10 Classification: TRANSFERASE Ligands: GDK, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-10
Ligands: GDK, GOL
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Crystal Structure Of Spleen Tyrosine Kinase (Syk) In Complex With A 2-(Phenoxymethyl)Pyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2018-10-10 Classification: TRANSFERASE Ligands: GDH, BR, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-10
Ligands: GDH, BR, GOL, DMS
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Human Spleen Tyrosine Kinase Kinase Domain In Complex With Azanaphthyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2016-09-14 Classification: TRANSFERASE Ligands: 6ZG, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: 6ZG, GOL, DMS
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Human Spleen Tyrosine Kinase Kinase Domain In Complex With Azanaphthyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2016-09-14 Classification: TRANSFERASE Ligands: 6ZF, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: 6ZF, GOL
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000222
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DF, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DF, GOL
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000223
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DL, DMS
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Syk Kinase Domain In Complex With Inhibitor Gtc000224
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.34 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DK
 |
Syk Kinase Domain In Complex With Inhibitor Gtc000225
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DJ
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000226
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.22 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DN
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000233
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: GOL, 4DQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: GOL, 4DQ
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The Kinase Domain Of Human Spleen Tyrosine (Syk) In Complex With Gtc000249
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: 4DO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: 4DO
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Crystal Structure Of Human Peptidylarginine Deiminase Type4 (Pad4) In Complex With Gsk147
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2015-01-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, 3YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: CA, 3YZ
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Crystal Structure Of Human Peptidylarginine Deiminase Type4 (Pad4) In Complex With Gsk199
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.29 Å Release Date: 2015-01-28 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CA, 3Z0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-01-28
Ligands: CA, 3Z0