Search Count: 93
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Hiv-1 Integrase Catalytic Core Domain Mutant (Kgd) In Complex With Inhibitor Grl-142
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2023-03-22 Classification: VIRAL PROTEIN Ligands: 7OA, SO4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: 7OA, SO4
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Crystal Structure Of Sars-Cov-2 Main Protease In Complex With An Inhibitor Grl-2420
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2020-09-23 Classification: VIRAL PROTEIN/INHIBITOR Ligands: V7G, 1PE |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: V7G, 1PE
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X-Ray Structure Of Sars-Cov-2 Main Protease Bound To Grl-024-20 At 1.45 A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2020-08-19 Classification: HYDROLASE Ligands: V7G |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2020-08-19
Ligands: V7G
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X-Ray Crystal Structure Of Wild Type Hiv-1 Protease In Complex With Grl-004
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2020-05-20 Classification: VIRAL PROTEIN/INHIBITOR Ligands: NKA |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-05-20
Ligands: NKA
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X-Ray Crystal Structure Of Wild Type Hiv-1 Protease In Complex With Grl-002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2020-05-20 Classification: VIRAL PROTEIN/INHIBITOR Ligands: NJY |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-05-20
Ligands: NJY
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X-Ray Crystal Structure Of Darunavir-Resistant Hiv-1 Protease (P51) In Complex With Grl-003
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.21 Å Release Date: 2020-04-08 Classification: VIRAL PROTEIN/INHIBITOR Ligands: GOL, EDO, JDV |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GOL, EDO, JDV
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X-Ray Crystal Structure Of Wild Type Hiv-1 Protease In Complex With Grl-063
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2020-04-08 Classification: VIRAL PROTEIN/INHIBITOR Ligands: EDO, MJD |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: EDO, MJD
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X-Ray Crystal Structure Of Darunavir-Resistant Hiv-1 Protease (P30) In Complex With Grl-003
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2020-04-08 Classification: VIRAL PROTEIN/INHIBITOR Ligands: GOL, PEG, JDV, SO4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GOL, PEG, JDV, SO4
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X-Ray Crystal Structure Of Darunavir-Resistant Hiv-1 Protease (P30) In Complex With Grl-001
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2020-04-08 Classification: VIRAL PROTEIN/INHIBITOR Ligands: PEG, GOL, JDY, SO4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: PEG, GOL, JDY, SO4
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X-Ray Crystal Structure Of Darunavir-Resistant Hiv-1 Protease (P51) In Complex With Grl-001
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.21 Å Release Date: 2020-04-08 Classification: VIRAL PROTEIN/INHIBITOR Ligands: GOL, JDY, EDO |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-04-08
Ligands: GOL, JDY, EDO
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Crystal Structure Of Biotin Acetyl Coenzyme A Carboxylase Synthetase From Helicobacter Pylori With Bound Biotinylated Atp
Organism: Helicobacter pylori (strain g27)
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-04-04 Classification: LIGASE Ligands: F5D, SO4, EDO |
Organism: Helicobacter pylori (strain g27)
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: F5D, SO4, EDO
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X-Ray Crystal Structure Of Wild Type Hiv-1 Protease In Complex With Grl-121
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7O7 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 7O7
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X-Ray Crystal Structure Of Wild Type Hiv-1 Protease In Complex With Grl-142
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2017-10-18 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 7OA |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2017-10-18
Ligands: 7OA
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Crystal Structure Of Multidrug-Resistant Clinical Isolate A02 Hiv-1 Protease In Complex With Non-Peptidic Inhibitor, Grl0519
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2016-05-04 Classification: hydrolase/hydrolase inhibitor Ligands: G52 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: G52
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Crystal Structure Of Multidrug-Resistant Clinical Isolate A02 Hiv-1 Protease In Complex With Amprenavir
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-05-04 Classification: hydrolase/hydrolase inhibitor Ligands: 478 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 478
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Crystal Structure Of Multidrug-Resistant Clinical Isolate A02 Hiv-1 Protease In Complex With Non-Peptidic Inhibitor, Grl079
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2016-05-04 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 79G |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 79G
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Crystal Structure Of Fab Fragment Of Monoclonal Antibody Roab13
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-06-24 Classification: IMMUNE SYSTEM |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-06-24
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Crystal Structure Of Btk Kinase Domain Complexed With 6-(Dimethylamino)-2-[2-(Hydroxymethyl)-3-[1-Methyl-5-[[5-(Morpholine-4-Carbonyl)-2-Pyridyl]Amino]-6-Oxo-3-Pyridyl]Phenyl]-3,4-Dihydroisoquinolin-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-12-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3OU, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3OU, DMS
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Crystal Structure Of Btk Kinase Domain Complexed With 6-(Dimethylamino)-8-Fluoro-2-[2-(Hydroxymethyl)-3-[1-Methyl-5-[[5-(Morpholine-4-Carbonyl)-2-Pyridyl]Amino]-6-Oxo-3-Pyridyl]Phenyl]Isoquinolin-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.17 Å Release Date: 2014-12-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3OV, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3OV, DMS
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Crystal Structure Of Btk Kinase Domain Complexed With 2-[8-Fluoro-2-[2-(Hydroxymethyl)-3-[1-Methyl-5-[[5-(4-Methylpiperazin-1-Yl)-2-Pyridyl]Amino]-6-Oxo-3-Pyridyl]Phenyl]-1-Oxo-3,4-Dihydroisoquinolin-6-Yl]-2-Methyl-Propanenitrile
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-12-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3P0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-24
Ligands: 3P0
