Search Count: 22
![]() |
X-Ray Studies Of Ku70/80 Reveal The Binding Site For Ip6
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:3.70 Å Release Date: 2023-08-30 Classification: DNA BINDING PROTEIN Ligands: IHP |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2023-08-30
Ligands: IHP
![]() |
Cryoem Structure Of Ku Heterodimer Bound To Dna
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-05-24 Classification: DNA BINDING PROTEIN Ligands: IHP |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-05-24
Ligands: IHP
![]() |
Cryo-Em Structure Of Ku 70/80 Bound To Inositol Hexakisphosphate
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2023-05-17 Classification: DNA BINDING PROTEIN Ligands: IHP |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2023-05-17
Ligands: IHP
![]() |
Estrogen Receptor Alpha In Complex With Compound 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2023-02-01 Classification: TRANSCRIPTION Ligands: H09 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: H09
![]() |
Oestrogen Receptor Ligand Binding Domain In Complex With Compound 38
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2023-02-01 Classification: GENE REGULATION Ligands: GZI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-02-01
Ligands: GZI
![]() |
Crystal Structure Of The Bromodomain Of Atad2 With Az13824374
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 96L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 96L
![]() |
Crystal Structure Of The Bromodomain Of Atad2 With Phenol Hts Hit (Cpd 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 963 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 963
![]() |
Crystal Structure Of The Bromodomain Of Atad2 With Triazolopyridine (Cpd 14)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 95O |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 95O
![]() |
Crystal Structure Of The Bromodomain Of Atad2 With Triazolopyridazine (Cpd 22)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.96 Å Release Date: 2022-01-19 Classification: GENE REGULATION Ligands: SO4, 93L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: SO4, 93L
![]() |
Crystal Structure Of Beta-Catenin In Complex With Cyclic Peptide Inhibitor
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-04-07 Classification: SIGNALING PROTEIN Ligands: EPE, CL |
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2021-04-07
Ligands: EPE, CL
![]() |
Oestrogen Receptor Ligand Binding Domain In Complex With Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNE
![]() |
Oestrogen Receptor Ligand Binding Domain In Complex With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNH
![]() |
Oestrogen Receptor Ligand Binding Domain In Complex With Compound 18
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-01-20 Classification: GENE REGULATION Ligands: QNK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: QNK
![]() |
Crystal Structure Of Mtead With A Vgl4 Tertiary Structure Mimetic
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2020-09-30 Classification: SIGNALING PROTEIN Ligands: GOL, ACE |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2020-09-30
Ligands: GOL, ACE
![]() |
Era_L536S (L536S/C381S/C471S,C530S) In Complex With A Bridged Tetracyclic Indole (Compound 8)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-10-30 Classification: GENE REGULATION Ligands: LRQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-30
Ligands: LRQ
![]() |
Era_L536S (L536S/C381S/C471S,C530S) In Complex With A Tricyclic Indole (Compound 6)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2019-10-30 Classification: GENE REGULATION Ligands: LVH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-30
Ligands: LVH
![]() |
Tricyclic Indazoles A Novel Class Of Selective Estrogen Receptor Degrader Antagonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2019-01-23 Classification: DNA BINDING PROTEIN Ligands: H8W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: H8W
![]() |
Crystal Structure Of The Bcl6 Btb Domain In Complex With Anilinopyrimidine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: C0H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: C0H
![]() |
Crystal Structure Of The Bcl6 Btb Domain In Complex With Anilinopyrimidine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: CL, C1W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: CL, C1W
![]() |
Crystal Structure Of The Bcl6 Btb Domain In Complex With Anilinopyrimidine Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2018-10-24 Classification: TRANSFERASE Ligands: CL, C0Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: CL, C0Q
